# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5082977 | 18 | INH | 0 | ALA5049259 | Active | % | Homo sapiens | ||||
2. | ALA5082977 | 18 | Activity | 0 | ALA5049258 | Active | ||||||
3. | ALA5082977 | 18 | Activity | 0 | ALA5049257 | Active | ||||||
4. | ALA5082977 | 18 | Activity | 0 | ALA5049256 | Active | ||||||
5. | ALA5082977 | 18 | Activity | 0 | ALA5049255 | Active | ||||||
6. | ALA5082977 | 18 | Activity | 0 | ALA5049254 | Active | ||||||
7. | ALA5082977 | 18 | Activity | 0 | ALA5049253 | Dose-Dependent Effect | ||||||
8. | ALA5082977 | 18 | Activity | 0 | ALA5049252 | Dose-Dependent Effect | ||||||
9. | ALA5082977 | 18 | Activity | 0 | ALA5049251 | Dose-Dependent Effect | ||||||
10. | ALA5082977 | 18 | Activity | 0 | ALA5049250 | Dose-Dependent Effect | ||||||
11. | ALA5082977 | 18 | Activity | 0 | ALA5049249 | Dose-Dependent Effect | ||||||
12. | ALA5082977 | 18 | IC50 | = | 100 | uM | ALA5049248 | 4.00 | nM | Homo sapiens | ||
13. | ALA5082977 | 18 | IC50 | = | 31 | uM | ALA5049247 | 4.51 | nM | Homo sapiens | ||
14. | ALA5082977 | 18 | IC50 | = | 98 | uM | ALA5049246 | 4.01 | nM | Homo sapiens | ||
15. | ALA5082977 | 18 | Kcat | = | 13.4 | /min | ALA5049245 | /min | Homo sapiens | |||
16. | ALA5082977 | 18 | K | = | 113 | uM | ALA5049244 | uM | Homo sapiens | |||
17. | ALA5082977 | 18 | Km | = | 2.82 | uM | ALA5049243 | nM | Homo sapiens | |||
18. | ALA5082977 | 18 | Ki | = | 0.3 | uM | ALA5049242 | 6.52 | nM | Homo sapiens | ||
19. | ALA5082977 | 18 | Activity | = | 4.21 | % | ALA5049241 | % | Homo sapiens | |||
20. | ALA5082977 | 18 | Activity | < | 15 | % | ALA5049238 | % | Homo sapiens |