# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5086057 | [64Cu]Cu-NODAGA-cLAB1-TATE | SUV | = | 1 | ALA5043882 | ||||||
2. | ALA5086057 | [64Cu]Cu-NODAGA-cLAB1-TATE | Drug uptake | = | 16 | % | ALA5043873 | % | ||||
3. | ALA5086057 | [64Cu]Cu-NODAGA-cLAB1-TATE | Drug uptake | = | 87 | % | ALA5043870 | % | ||||
4. | ALA5086057 | [64Cu]Cu-NODAGA-cLAB1-TATE | t1/2 | 0 | ALA5043869 | Not Determined | ||||||
5. | ALA5086057 | [64Cu]Cu-NODAGA-cLAB1-TATE | t1/2 | 0 | ALA5043868 | Not Determined | ||||||
6. | ALA5086057 | [64Cu]Cu-NODAGA-cLAB1-TATE | Bmax | = | 1190 | fmol/mg | ALA5043867 | fmol/mg | Mus musculus | |||
7. | ALA5086057 | [64Cu]Cu-NODAGA-cLAB1-TATE | Kd | = | 8.57 | nM | ALA5043866 | 8.07 | nM | Mus musculus | ||
8. | ALA5086057 | [64Cu]Cu-NODAGA-cLAB1-TATE | Kd | = | 3.1 | uM | ALA5043865 | 5.51 | nM | Homo sapiens | ||
9. | ALA5086057 | [64Cu]Cu-NODAGA-cLAB1-TATE | logD | = | -1.49 | ALA5043864 | ||||||
10. | ALA5086057 | [64Cu]Cu-NODAGA-cLAB1-TATE | PB | < | 30 | % | ALA5043863 | % | Homo sapiens | |||
11. | ALA5086057 | [64Cu]Cu-NODAGA-cLAB1-TATE | PPB | = | 46 | % | ALA5043862 | % |