| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5086545 | 12 | Ratio | = | 0.75 | ALA5042450 | ||||||
| 2. | ALA5086545 | 12 | Papp | = | 0.915 | 10^-6 cm/s | ALA5042449 | 10^-6 cm/s | ||||
| 3. | ALA5086545 | 12 | Papp | = | 1.22 | 10^-6 cm/s | ALA5042448 | 10^-6 cm/s | ||||
| 4. | ALA5086545 | 12 | t1/2 | = | 192 | min | ALA5042447 | hr | ||||
| 5. | ALA5086545 | 12 | CLH | = | 6.48 | ml/min.kg | ALA5042446 | mL.min-1.kg-1 | ||||
| 6. | ALA5086545 | 12 | INH | = | 5.1 | % | ALA5042445 | % | Homo sapiens | |||
| 7. | ALA5086545 | 12 | IC50 | = | 1039 | nM | ALA5042444 | 5.98 | nM | Homo sapiens | ||
| 8. | ALA5086545 | 12 | IC50 | = | 60 | nM | ALA5042443 | 7.22 | nM | Homo sapiens | ||
| 9. | ALA5086545 | 12 | solubility | = | 77 | uM | ALA5042442 | nM | ||||
| 10. | ALA5086545 | 12 | solubility | > | 100 | uM | ALA5042441 | nM | ||||
| 11. | ALA5086545 | 12 | Ki | = | 813 | nM | ALA5042440 | 6.09 | nM | Homo sapiens | ||
| 12. | ALA5086545 | 12 | Ki | = | 885 | nM | ALA5042439 | 6.05 | nM | Homo sapiens | ||
| 13. | ALA5086545 | 12 | Ki | > | 10000 | nM | ALA5042438 | nM | Homo sapiens | |||
| 14. | ALA5086545 | 12 | Ki | = | 125 | nM | ALA5042437 | 6.90 | nM | Homo sapiens | ||
| 15. | ALA5086545 | 12 | Ki | > | 10000 | nM | ALA5042436 | nM | Homo sapiens |
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