| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5088381 | SY-5102 | Activity | 0 | ALA5043168 | Dose-Dependent Effect | Homo sapiens | |||||
| 2. | ALA5088381 | SY-5102 | IC50 | = | 75 | nM | ALA5043166 | 7.12 | nM | Homo sapiens | ||
| 3. | ALA5088381 | SY-5102 | IC50 | = | 90 | nM | ALA5043165 | 7.05 | nM | Homo sapiens | ||
| 4. | ALA5088381 | SY-5102 | Kd | = | 0.03 | nM | ALA5043164 | 10.52 | nM | Homo sapiens | ||
| 5. | ALA5088381 | SY-5102 | EC50 | = | 9 | nM | ALA5043163 | 8.05 | nM | Homo sapiens | ||
| 6. | ALA5088381 | SY-5102 | IC50 | = | 189 | nM | ALA5043162 | 6.72 | nM | Homo sapiens | ||
| 7. | ALA5088381 | SY-5102 | logD | = | 2.6 | ALA5043160 | ||||||
| 8. | ALA5088381 | SY-5102 | CLH | < | 38 | ml/min.kg | ALA5043159 | mL.min-1.kg-1 | ||||
| 9. | ALA5088381 | SY-5102 | Papp | = | 4.62 | 10^-6 cm/s | ALA5043158 | 10^-6 cm/s | ||||
| 10. | ALA5088381 | SY-5102 | CL free | = | 712 | ml/min.kg | ALA5043157 | mL.min-1.kg-1 | ||||
| 11. | ALA5088381 | SY-5102 | F | = | 36 | % | ALA5043156 | % | ||||
| 12. | ALA5088381 | SY-5102 | Activity | 0 | ALA5043155 | Active | Homo sapiens |
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