| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5089071 | 1 | Activity | 0 | ALA5050317 | Active | Trypanosoma congolense | |||||
| 2. | ALA5089071 | 1 | EC50 | 0 | ALA5050305 | Not Determined | Rattus norvegicus | |||||
| 3. | ALA5089071 | 1 | AUC | = | 21000 | ng.min/ml | ALA5050302 | ng.hr.mL-1 | ||||
| 4. | ALA5089071 | 1 | Cmax | = | 130 | ng/ml | ALA5050301 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 5. | ALA5089071 | 1 | AUC | = | 130000 | ng.min/ml | ALA5050299 | ng.hr.mL-1 | ||||
| 6. | ALA5089071 | 1 | t1/2 | = | 1.8 | hr | ALA5050297 | hr | ||||
| 7. | ALA5089071 | 1 | Vdss | = | 2.4 | L/Kg | ALA5050295 | L.kg-1 | ||||
| 8. | ALA5089071 | 1 | CL | = | 20 | ml/min.kg | ALA5050293 | mL.min-1.kg-1 | ||||
| 9. | ALA5089071 | 1 | Activity | = | 100 | % | ALA5050292 | % | Trypanosoma vivax | |||
| 10. | ALA5089071 | 1 | Activity | = | 100 | % | ALA5050291 | % | Trypanosoma vivax | |||
| 11. | ALA5089071 | 1 | Activity | = | 100 | % | ALA5050290 | % | Trypanosoma vivax | |||
| 12. | ALA5089071 | 1 | Activity | = | 100 | % | ALA5050289 | % | Trypanosoma congolense | |||
| 13. | ALA5089071 | 1 | Activity | = | 100 | % | ALA5050288 | % | Trypanosoma congolense | |||
| 14. | ALA5089071 | 1 | Activity | = | 100 | % | ALA5050287 | % | Trypanosoma brucei brucei | |||
| 15. | ALA5089071 | 1 | t1/2 | = | 1 | hr | ALA5050286 | hr | ||||
| 16. | ALA5089071 | 1 | F | = | 74 | % | ALA5050285 | % | ||||
| 17. | ALA5089071 | 1 | MTD | > | 300 | mg kg-1 | ALA5050284 | mg kg-1 | ||||
| 18. | ALA5089071 | 1 | Fu | = | 0.16 | % | ALA5050283 | |||||
| 19. | ALA5089071 | 1 | CLH | = | 0.5 | ml/min/g | ALA5050282 | mL.min-1.g-1 | ||||
| 20. | ALA5089071 | 1 | CLH | < | 0.5 | ml/min/g | ALA5050281 | mL.min-1.g-1 |
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