| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5089544 | 46; AGB1 | Emax | = | 97 | % | ALA5054796 | % | Homo sapiens | |||
| 2. | ALA5089544 | 46; AGB1 | pDC50 | = | 7.9 | ALA5054795 | Homo sapiens | |||||
| 3. | ALA5089544 | 46; AGB1 | F | = | 140 | % | ALA5054793 | % | ||||
| 4. | ALA5089544 | 46; AGB1 | Cmax | = | 0.7 | uM | ALA5054792 | nM | ||||
| 5. | ALA5089544 | 46; AGB1 | Tmax | = | 0.5 | hr | ALA5054791 | hr | ||||
| 6. | ALA5089544 | 46; AGB1 | MRT | = | 0.39 | hr | ALA5054790 | hr | ||||
| 7. | ALA5089544 | 46; AGB1 | AUC | = | 2.4 | uM.hr | ALA5054789 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 8. | ALA5089544 | 46; AGB1 | AUC | = | 1.72 | uM.hr | ALA5054788 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 9. | ALA5089544 | 46; AGB1 | AUClast | = | 2.33 | uM.hr | ALA5054787 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 10. | ALA5089544 | 46; AGB1 | AUClast | = | 1.71 | uM.hr | ALA5054786 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 11. | ALA5089544 | 46; AGB1 | t1/2 | = | 1.65 | hr | ALA5054785 | hr | ||||
| 12. | ALA5089544 | 46; AGB1 | t1/2 | = | 1.49 | hr | ALA5054784 | hr | ||||
| 13. | ALA5089544 | 46; AGB1 | Vdss | = | 1.1 | L/Kg | ALA5054783 | L.kg-1 | ||||
| 14. | ALA5089544 | 46; AGB1 | CL | = | 47.2 | ml/min.kg | ALA5054782 | mL.min-1.kg-1 | ||||
| 15. | ALA5089544 | 46; AGB1 | Stability | 0 | ALA5054781 | Stable | % | |||||
| 16. | ALA5089544 | 46; AGB1 | INH | 0 | ALA5054780 | Active | % | |||||
| 17. | ALA5089544 | 46; AGB1 | INH | 0 | ALA5054779 | Active | % | |||||
| 18. | ALA5089544 | 46; AGB1 | INH | 0 | ALA5054778 | Active | % | |||||
| 19. | ALA5089544 | 46; AGB1 | pEC50 | = | 7.6 | ALA5054775 | 7.60 | nM | Homo sapiens | |||
| 20. | ALA5089544 | 46; AGB1 | Kd | = | 11 | nM | ALA5054774 | 7.96 | nM |
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