| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5089882 | 7l | Activity | 0 | ALA5056459 | Active | ||||||
| 2. | ALA5089882 | 7l | Activity | 0 | ALA5056458 | Active | ||||||
| 3. | ALA5089882 | 7l | Activity | 0 | ALA5056457 | Active | ||||||
| 4. | ALA5089882 | 7l | INH | 0 | ALA5056456 | Active | % | Homo sapiens | ||||
| 5. | ALA5089882 | 7l | INH | 0 | ALA5056455 | Active | % | Homo sapiens | ||||
| 6. | ALA5089882 | 7l | Activity | 0 | ALA5056453 | Active | ||||||
| 7. | ALA5089882 | 7l | Selectivity Index | = | 1.3 | ALA5056452 | ||||||
| 8. | ALA5089882 | 7l | Activity | 0 | ALA5056451 | Active | Homo sapiens | |||||
| 9. | ALA5089882 | 7l | IC50 | = | 0.95 | uM | ALA5056450 | 6.02 | nM | Rattus norvegicus | ||
| 10. | ALA5089882 | 7l | IC50 | = | 1.2 | uM | ALA5056449 | 5.92 | nM | Rattus norvegicus | ||
| 11. | ALA5089882 | 7l | solubility | = | 195.8 | uM | ALA5056448 | nM | ||||
| 12. | ALA5089882 | 7l | Papp | = | 44.1 | 10^-6 cm/s | ALA5056447 | 10^-6 cm/s | ||||
| 13. | ALA5089882 | 7l | Papp | = | 19.4 | 10^-6 cm/s | ALA5056446 | 10^-6 cm/s | ||||
| 14. | ALA5089882 | 7l | CLH | = | 58.3 | uL | ALA5056445 | uL | ||||
| 15. | ALA5089882 | 7l | t1/2 | = | 118.9 | min | ALA5056444 | hr | ||||
| 16. | ALA5089882 | 7l | IC50 | = | 0.18 | uM | ALA5056443 | 6.75 | nM | Homo sapiens | ||
| 17. | ALA5089882 | 7l | IC50 | = | 2.5 | uM | ALA5056442 | 5.60 | nM | Homo sapiens | ||
| 18. | ALA5089882 | 7l | INH | = | 5.7 | uM | ALA5056441 | uM | Homo sapiens | |||
| 19. | ALA5089882 | 7l | INH | > | 60 | % | ALA5056439 | % | Homo sapiens | |||
| 20. | ALA5089882 | 7l | INH | > | 60 | % | ALA5056438 | % | Homo sapiens |
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