| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  Kumatakenin | 22 | GI | = | 25.2 | % | ALA3412097 | % | Trypanosoma brucei gambiense | |||
| 2. | Kumatakenin | 22 | GI | = | 26.4 | % | ALA3412096 | % | Trypanosoma brucei gambiense | |||
| 3. | Kumatakenin | 22 | GI | = | 7.2 | % | ALA3412094 | % | Plasmodium falciparum | |||
| 4. | Kumatakenin | 22 | IC50 | = | 22.95 | uM | ALA3412093 | 4.64 | nM | Leishmania amazonensis | ||
| 5. | Kumatakenin | 22 | Activity | = | 50 | uM | ALA3412090 | uM | ||||
| 6. | Kumatakenin | 22 | IC50 | = | 57.5 | uM | ALA3412089 | 4.24 | nM | Mus musculus | ||
| 7. | Kumatakenin | 22 | Activity | = | 81.3 | % | ALA3412088 | % | Rattus norvegicus | |||
| 8. | Kumatakenin | 22 | Activity | = | 38.7 | % | ALA3412087 | % | Rattus norvegicus | |||
| 9. | Kumatakenin | 22 | IC50 | = | 10.3 | uM | ALA4343927 | 4.99 | nM | Homo sapiens | ||
| 10. | Kumatakenin | 22 | IC50 | = | 8.1 | uM | ALA4343926 | 5.09 | nM | Homo sapiens | ||
| 11. | Kumatakenin | 22 | INH | > | 40 | % | ALA4612144 | % | ||||
| 12. | Kumatakenin | 22 | Activity | = | 80 | % | ALA4612145 | % | Homo sapiens | |||
| 13. | Kumatakenin | 22 | INH | > | 60 | % | ALA4612143 | % | Homo sapiens | |||
| 14. | Kumatakenin | 22 | IC50 | = | 0.7 | ug ml-1 | ALA930440 | ug.mL-1 | ||||
| 15. | Kumatakenin | 22 | IC50 | = | 1.2 | ug ml-1 | ALA930438 | ug.mL-1 | ||||
| 16. | Kumatakenin | 22 | Ki | = | 90.3 | uM | ALA1073435 | 4.04 | nM | |||
| 17. | Kumatakenin | 22 | IC50 | = | 36.4 | uM | ALA1073434 | 4.44 | nM | |||
| 18. | Kumatakenin | 22 | Therapeutic index 99 | = | 40 | ALA851082 | ||||||
| 19. | Kumatakenin | 22 | Therapeutic index 99 | = | 333.3 | ALA851081 | ||||||
| 20. | Kumatakenin | 22 | ED99 | = | 2.5 | ug ml-1 | ALA799318 | ug ml-1 | Human rhinovirus sp. |
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