| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5091040 | 17 | Activity | 0 | ALA5035833 | Not Active | ||||||
| 2. | ALA5091040 | 17 | CL free | = | 453 | ml/min.kg | ALA5035815 | mL.min-1.kg-1 | ||||
| 3. | ALA5091040 | 17 | EC50 | = | 130 | nM | ALA5035814 | 6.89 | nM | Homo sapiens | ||
| 4. | ALA5091040 | 17 | PB | = | 99 | % | ALA5035813 | % | ||||
| 5. | ALA5091040 | 17 | t1/2 | = | 3.9 | hr | ALA5035812 | hr | ||||
| 6. | ALA5091040 | 17 | Vdss | = | 0.9 | L/Kg | ALA5035811 | L.kg-1 | ||||
| 7. | ALA5091040 | 17 | CL | = | 4.4 | ml/min.kg | ALA5035810 | mL.min-1.kg-1 | ||||
| 8. | ALA5091040 | 17 | AUC | = | 2921.5 | nM.hr | ALA5035809 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 9. | ALA5091040 | 17 | CL free | = | 576 | ml/min.kg | ALA5035808 | mL.min-1.kg-1 | ||||
| 10. | ALA5091040 | 17 | PB | = | 97.6 | % | ALA5035807 | % | ||||
| 11. | ALA5091040 | 17 | t1/2 | = | 3.4 | hr | ALA5035806 | hr | ||||
| 12. | ALA5091040 | 17 | Vdss | = | 2.1 | L/Kg | ALA5035805 | L.kg-1 | ||||
| 13. | ALA5091040 | 17 | CL | = | 19.6 | ml/min.kg | ALA5035804 | mL.min-1.kg-1 | ||||
| 14. | ALA5091040 | 17 | AUC | = | 647.9 | nM.hr | ALA5035803 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 15. | ALA5091040 | 17 | CL free | > | 3000 | ml/min.kg | ALA5035802 | mL.min-1.kg-1 | ||||
| 16. | ALA5091040 | 17 | PB | = | 99 | % | ALA5035801 | % | ||||
| 17. | ALA5091040 | 17 | t1/2 | = | 2.1 | hr | ALA5035800 | hr | ||||
| 18. | ALA5091040 | 17 | Vdss | = | 0.8 | L/Kg | ALA5035799 | L.kg-1 | ||||
| 19. | ALA5091040 | 17 | CL | = | 28.7 | ml/min.kg | ALA5035798 | mL.min-1.kg-1 | ||||
| 20. | ALA5091040 | 17 | AUC | = | 441.7 | nM.hr | ALA5035797 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 |
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