| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5092315 | 9ka | INH | 0 | ALA5048566 | Dose-Dependent Effect | % | |||||
| 2. | ALA5092315 | 9ka | Activity | 0 | ALA5048565 | Non-Toxic | ||||||
| 3. | ALA5092315 | 9ka | Activity | 0 | ALA5048564 | Non-Toxic | ||||||
| 4. | ALA5092315 | 9ka | TGI | = | 95.19 | % | ALA5048563 | % | Homo sapiens | |||
| 5. | ALA5092315 | 9ka | Activity | 0 | ALA5048562 | Active | Homo sapiens | |||||
| 6. | ALA5092315 | 9ka | Activity | 0 | ALA5048561 | Active | Homo sapiens | |||||
| 7. | ALA5092315 | 9ka | Activity | 0 | ALA5048560 | Active | Homo sapiens | |||||
| 8. | ALA5092315 | 9ka | Activity | 0 | ALA5048559 | Active | Homo sapiens | |||||
| 9. | ALA5092315 | 9ka | Kd | = | 6.2 | nM | ALA5048558 | 8.21 | nM | Homo sapiens | ||
| 10. | ALA5092315 | 9ka | INH | 0 | ALA5048557 | Dose-Dependent Effect | % | |||||
| 11. | ALA5092315 | 9ka | INH | 0 | ALA5048556 | Dose-Dependent Effect | % | |||||
| 12. | ALA5092315 | 9ka | F | = | 50.97 | % | ALA5048555 | % | ||||
| 13. | ALA5092315 | 9ka | CL | = | 6.15 | ml/min.kg | ALA5048554 | mL.min-1.kg-1 | ||||
| 14. | ALA5092315 | 9ka | AUCt | = | 38950.06 | hr.ng/ml | ALA5048553 | ng.hr.mL-1 | ||||
| 15. | ALA5092315 | 9ka | AUCt | = | 15282.64 | hr.ng/ml | ALA5048552 | ng.hr.mL-1 | ||||
| 16. | ALA5092315 | 9ka | Cmax | = | 8558.59 | ng/ml | ALA5048551 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 17. | ALA5092315 | 9ka | Cmax | = | 11085.51 | ng/ml | ALA5048550 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 18. | ALA5092315 | 9ka | t1/2 | = | 3.06 | hr | ALA5048549 | hr | ||||
| 19. | ALA5092315 | 9ka | t1/2 | = | 0.89 | hr | ALA5048548 | hr | ||||
| 20. | ALA5092315 | 9ka | INH | = | 10 | % | ALA5048547 | % | Homo sapiens |
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