# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5092617 | 8 | F | = | 98 | % | ALA5036648 | % | ||||
2. | ALA5092617 | 8 | AUC | = | 3766 | hr.ng/ml | ALA5036647 | ng.hr.mL-1 | ||||
3. | ALA5092617 | 8 | Cmax | = | 995 | ng/ml | ALA5036646 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
4. | ALA5092617 | 8 | t1/2 | = | 2.6 | hr | ALA5036645 | hr | ||||
5. | ALA5092617 | 8 | Stability | = | 56 | % | ALA5036644 | % | ||||
6. | ALA5092617 | 8 | IC50 | = | 3.2 | nM | ALA5036643 | 8.49 | nM | Homo sapiens | ||
7. | ALA5092617 | 8 | GI90 | = | 43 | nM | ALA5036642 | nM | Homo sapiens | |||
8. | ALA5092617 | 8 | GI50 | = | 3 | nM | ALA5036642 | nM | Homo sapiens | |||
9. | ALA5092617 | 8 | deltaTm | = | 16.1 | degrees C | ALA5036641 | degrees C | Homo sapiens |