| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5092744 | L7 | Kd | = | 3.34 | nM | ALA5225070 | 8.48 | nM | Homo sapiens | ||
| 2. | ALA5092744 | L7 | RLU | = | 1.81 | ALA5033028 | Homo sapiens | |||||
| 3. | ALA5092744 | L7 | IC50 | > | 30 | uM | ALA5032997 | nM | Homo sapiens | |||
| 4. | ALA5092744 | L7 | F | = | 0.35 | % | ALA5032977 | % | ||||
| 5. | ALA5092744 | L7 | AUCt | = | 15.2 | hr.ng/ml | ALA5032976 | ng.hr.mL-1 | ||||
| 6. | ALA5092744 | L7 | Cmax | = | 4.46 | ng/ml | ALA5032975 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 7. | ALA5092744 | L7 | Tmax | = | 2.33 | hr | ALA5032974 | hr | ||||
| 8. | ALA5092744 | L7 | t1/2 | = | 4.17 | hr | ALA5032973 | hr | ||||
| 9. | ALA5092744 | L7 | CL | = | 2377 | ml/hr/kg | ALA5032972 | mL.min-1.kg-1 | ||||
| 10. | ALA5092744 | L7 | AUCt | = | 860 | hr.ng/ml | ALA5032971 | ng.hr.mL-1 | ||||
| 11. | ALA5092744 | L7 | Cmax | = | 2087 | ng/ml | ALA5032970 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 12. | ALA5092744 | L7 | Tmax | = | 0.08 | hr | ALA5032969 | hr | ||||
| 13. | ALA5092744 | L7 | t1/2 | = | 4.04 | hr | ALA5032968 | hr | ||||
| 14. | ALA5092744 | L7 | EC50 | = | 375 | nM | ALA5032967 | 6.43 | nM | Homo sapiens | ||
| 15. | ALA5092744 | L7 | Activity | 0 | ALA5032963 | Not Active | Mus musculus | |||||
| 16. | ALA5092744 | L7 | Activity | 0 | ALA5032962 | Not Active | Cricetulus griseus | |||||
| 17. | ALA5092744 | L7 | Activity | 0 | ALA5032961 | Not Active | Homo sapiens | |||||
| 18. | ALA5092744 | L7 | Kd | = | 3.34 | nM | ALA5032960 | 8.48 | nM | Homo sapiens | ||
| 19. | ALA5092744 | L7 | Activity | 0 | ALA5032959 | Not Active | Homo sapiens | |||||
| 20. | ALA5092744 | L7 | IC50 | = | 1.8 | nM | ALA5032958 | 8.74 | nM | Homo sapiens |
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