| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5169772 | X4 | Activity | 0 | ALA5153823 | NA | Mus musculus | |||||
| 2. | ALA5169772 | X4 | IC50 | > | 50 | uM | ALA5153822 | nM | Mus musculus | |||
| 3. | ALA5169772 | X4 | F | = | 2.3 | % | ALA5153810 | % | ||||
| 4. | ALA5169772 | X4 | CL | = | 3.5 | L/hr/kg | ALA5153808 | mL.min-1.kg-1 | ||||
| 5. | ALA5169772 | X4 | AUC | = | 582.7 | hr.ng/ml | ALA5153806 | ng.hr.mL-1 | ||||
| 6. | ALA5169772 | X4 | AUC | = | 71.2 | hr.ng/ml | ALA5153805 | ng.hr.mL-1 | ||||
| 7. | ALA5169772 | X4 | Cmax | = | 1311.2 | ng/ml | ALA5153803 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 8. | ALA5169772 | X4 | Cmax | = | 16.3 | ng/ml | ALA5153802 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 9. | ALA5169772 | X4 | Tmax | = | 0.1 | hr | ALA5153800 | hr | ||||
| 10. | ALA5169772 | X4 | Tmax | = | 1.4 | hr | ALA5153799 | hr | ||||
| 11. | ALA5169772 | X4 | t1/2 | = | 7.8 | hr | ALA5153797 | hr | ||||
| 12. | ALA5169772 | X4 | t1/2 | = | 8.9 | hr | ALA5153796 | hr | ||||
| 13. | ALA5169772 | X4 | t1/2 | >= | 140 | min | ALA5153795 | hr | ||||
| 14. | ALA5169772 | X4 | Ratio | = | 12.25 | ALA5153794 | ||||||
| 15. | ALA5169772 | X4 | Papp | = | 4.34 | 10^-6 cm/s | ALA5153793 | 10^-6 cm/s | ||||
| 16. | ALA5169772 | X4 | Papp | = | 0.35 | 10^-6 cm/s | ALA5153792 | 10^-6 cm/s | ||||
| 17. | ALA5169772 | X4 | t1/2 | = | 264 | min | ALA5153791 | hr | ||||
| 18. | ALA5169772 | X4 | Kd | = | 127.7 | nM | ALA5153790 | 6.89 | nM | Homo sapiens | ||
| 19. | ALA5169772 | X4 | INH | 0 | ALA5153787 | NA | % | Homo sapiens | ||||
| 20. | ALA5169772 | X4 | INH | 0 | ALA5153786 | NA | % | Homo sapiens |
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