# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5170047 | 12b; EML709 | Time | = | 66.7 | s | ALA5138966 | hr | Homo sapiens | |||
2. | ALA5170047 | 12b; EML709 | K | = | 0.015 | 1/s | ALA5138965 | 1/s | Homo sapiens | |||
3. | ALA5170047 | 12b; EML709 | K | = | 6.52 | 10^3/Ms | ALA5138964 | 10^3/Ms | Homo sapiens | |||
4. | ALA5170047 | 12b; EML709 | Kd | = | 2300 | nM | ALA5138963 | 5.64 | nM | Homo sapiens | ||
5. | ALA5170047 | 12b; EML709 | Selectivity Index | = | 9 | ALA5138956 | ||||||
6. | ALA5170047 | 12b; EML709 | Selectivity Index | = | 0.26 | ALA5138955 | ||||||
7. | ALA5170047 | 12b; EML709 | Selectivity Index | > | 47 | ALA5138954 | ||||||
8. | ALA5170047 | 12b; EML709 | Selectivity Index | = | 36 | ALA5138953 | ||||||
9. | ALA5170047 | 12b; EML709 | Selectivity Index | = | 20 | ALA5138952 | ||||||
10. | ALA5170047 | 12b; EML709 | Selectivity Index | = | 5 | ALA5138951 | ||||||
11. | ALA5170047 | 12b; EML709 | IC50 | = | 18.68 | uM | ALA5138950 | 4.73 | nM | Homo sapiens | ||
12. | ALA5170047 | 12b; EML709 | IC50 | = | 0.55 | uM | ALA5138949 | 6.26 | nM | Homo sapiens | ||
13. | ALA5170047 | 12b; EML709 | IC50 | > | 100 | uM | ALA5138948 | nM | Homo sapiens | |||
14. | ALA5170047 | 12b; EML709 | IC50 | = | 76.7 | uM | ALA5138947 | 4.12 | nM | Homo sapiens | ||
15. | ALA5170047 | 12b; EML709 | IC50 | = | 2.14 | uM | ALA5138946 | 5.67 | nM | Homo sapiens | ||
16. | ALA5170047 | 12b; EML709 | IC50 | = | 43.41 | uM | ALA5138945 | 4.36 | nM | Homo sapiens | ||
17. | ALA5170047 | 12b; EML709 | IC50 | = | 11.67 | uM | ALA5138944 | 4.93 | nM | Homo sapiens | ||
18. | ALA5170047 | 12b; EML709 | Activity | = | 0.43 | % | ALA5138942 | % | Homo sapiens |