| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5170475 | 4 | Ki | = | 4.1 | 10^4/M | ALA5159127 | 10^4/M | Homo sapiens | |||
| 2. | ALA5170475 | 4 | Drug uptake | 0 | ALA5159126 | Active | ||||||
| 3. | ALA5170475 | 4 | Drug uptake | = | 7 | % | ALA5159125 | % | ||||
| 4. | ALA5170475 | 4 | Drug uptake | = | 25.5 | % | ALA5159124 | % | ||||
| 5. | ALA5170475 | 4 | Drug uptake | = | 20.9 | % | ALA5159123 | % | ||||
| 6. | ALA5170475 | 4 | Activity | 0 | ALA5159122 | NA | Homo sapiens | |||||
| 7. | ALA5170475 | 4 | Activity | 0 | ALA5159121 | NA | Homo sapiens | |||||
| 8. | ALA5170475 | 4 | deltaTm | = | 10 | degrees C | ALA5159120 | degrees C | Homo sapiens | |||
| 9. | ALA5170475 | 4 | Selectivity Index | = | 30 | ALA5159119 | ||||||
| 10. | ALA5170475 | 4 | Selectivity Index | = | 2.3 | ALA5159118 | ||||||
| 11. | ALA5170475 | 4 | Selectivity Index | = | 3.8 | ALA5159117 | ||||||
| 12. | ALA5170475 | 4 | IC50 | = | 1.8 | uM | ALA5159116 | 5.75 | nM | Homo sapiens | ||
| 13. | ALA5170475 | 4 | IC50 | = | 0.48 | uM | ALA5159115 | 6.32 | nM | Homo sapiens | ||
| 14. | ALA5170475 | 4 | IC50 | = | 0.8 | uM | ALA5159114 | 6.10 | nM | Leishmania major | ||
| 15. | ALA5170475 | 4 | IC50 | = | 0.06 | uM | ALA5159113 | 7.22 | nM | Trypanosoma brucei | ||
| 16. | ALA5170475 | 4 | Drug uptake | 0 | ALA5159112 | Active | ||||||
| 17. | ALA5170475 | 4 | Drug uptake | 0 | ALA5159111 | Active |
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