# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5171168 | 39 | INH | = | 71.78 | % | ALA5115675 | % | Mus musculus | |||
2. | ALA5171168 | 39 | INH | = | 41.97 | % | ALA5115674 | % | Mus musculus | |||
3. | ALA5171168 | 39 | Activity | 0 | ALA5115672 | Active | Mus musculus | |||||
4. | ALA5171168 | 39 | Activity | 0 | ALA5115671 | NA | Mus musculus | |||||
5. | ALA5171168 | 39 | INH | 0 | ALA5115669 | Active | % | |||||
6. | ALA5171168 | 39 | BPR | = | 0.2 | ALA5115665 | ||||||
7. | ALA5171168 | 39 | AUClast | = | 0.59 | hr.microg/ml | ALA5115664 | ng.hr.mL-1 | ||||
8. | ALA5171168 | 39 | AUClast | = | 2.96 | hr.microg/ml | ALA5115663 | ng.hr.mL-1 | ||||
9. | ALA5171168 | 39 | AUC | = | 5.21 | hr.microg/ml | ALA5115662 | ng.hr.mL-1 | ||||
10. | ALA5171168 | 39 | AUCt | = | 4.98 | hr.microg/ml | ALA5115661 | ng.hr.mL-1 | ||||
11. | ALA5171168 | 39 | t1/2 | = | 1.53 | hr | ALA5115660 | hr | ||||
12. | ALA5171168 | 39 | Cmax | = | 3.2 | ug ml-1 | ALA5115659 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
13. | ALA5171168 | 39 | Tmax | = | 0.36 | hr | ALA5115658 | hr | ||||
14. | ALA5171168 | 39 | logPeff | = | 4.4 | ALA5115657 | ||||||
15. | ALA5171168 | 39 | Activity | = | 110.8 | % | ALA5115656 | % | Mus musculus | |||
16. | ALA5171168 | 39 | INH | = | 92.4 | % | ALA5115655 | % | Homo sapiens | |||
17. | ALA5171168 | 39 | IC50 | = | 0.04 | uM | ALA5115654 | 7.40 | nM | Homo sapiens | ||
18. | ALA5171168 | 39 | INH | = | 98.4 | % | ALA5115653 | % | Homo sapiens |