# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5171732 | 3 | INH | = | 17 | % | ALA5157675 | % | ||||
2. | ALA5171732 | 3 | F | = | 0.1 | % | ALA5157674 | % | ||||
3. | ALA5171732 | 3 | MRT | = | 5.25 | hr | ALA5157673 | hr | ||||
4. | ALA5171732 | 3 | AUC | = | 2.62 | ng.hr/ml | ALA5157672 | ng.hr.mL-1 | ||||
5. | ALA5171732 | 3 | AUCt | = | 0.665 | ng.hr/ml | ALA5157671 | ng.hr.mL-1 | ||||
6. | ALA5171732 | 3 | t1/2 | = | 3.53 | hr | ALA5157670 | hr | ||||
7. | ALA5171732 | 3 | Cmax | = | 0.444 | ng/ml | ALA5157669 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
8. | ALA5171732 | 3 | Ct | < | 1.5 | ng/g | ALA5157668 | ng/g | ||||
9. | ALA5171732 | 3 | Cp | < | 0.3 | ng/ml | ALA5157667 | ng/ml | ||||
10. | ALA5171732 | 3 | solubility | = | 122 | uM | ALA5157659 | nM | ||||
11. | ALA5171732 | 3 | IC50 | = | 64 | nM | ALA5157658 | 7.19 | nM | Homo sapiens | ||
12. | ALA5171732 | 3 | permeability | < | 0.025 | 10^-6 cm/s | ALA5157657 | 10^-6 cm/s | ||||
13. | ALA5171732 | 3 | FaFg | = | 0.1 | % | ALA5109478 | % | ||||
14. | ALA5171732 | 3 | IC50 | = | 64 | nM | ALA5109473 | 7.19 | nM | Homo sapiens |