# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5172262 | 24 | Activity | 0 | ALA5144067 | Dde | Homo sapiens | |||||
2. | ALA5172262 | 24 | ED50 | < | 40 | mg kg-1 | ALA5144066 | mg.kg-1 | Homo sapiens | |||
3. | ALA5172262 | 24 | Activity | 0 | ALA5144065 | Toxic | ||||||
4. | ALA5172262 | 24 | TGI | = | 77.7 | % | ALA5144064 | % | Homo sapiens | |||
5. | ALA5172262 | 24 | Activity | = | 0.009 | g | ALA5144063 | g | Homo sapiens | |||
6. | ALA5172262 | 24 | Activity | = | 67 | mm3 | ALA5144062 | mm3 | Homo sapiens | |||
7. | ALA5172262 | 24 | Activity | = | 87 | mm3 | ALA5144061 | mm3 | Homo sapiens | |||
8. | ALA5172262 | 24 | Activity | = | 105 | mm3 | ALA5144060 | mm3 | Homo sapiens | |||
9. | ALA5172262 | 24 | Activity | = | 126 | mm3 | ALA5144059 | mm3 | Homo sapiens | |||
10. | ALA5172262 | 24 | Activity | = | 136 | mm3 | ALA5144058 | mm3 | Homo sapiens | |||
11. | ALA5172262 | 24 | Cp | = | 279 | ng/ml | ALA5144057 | ng/ml | ||||
12. | ALA5172262 | 24 | Time | = | 480 | min | ALA5144056 | hr | ||||
13. | ALA5172262 | 24 | beta t1/2 | = | 954.1 | min | ALA5144055 | hr | ||||
14. | ALA5172262 | 24 | AUC | = | 187.7 | ug/ml.min | ALA5144054 | ng.hr.mL-1 | ||||
15. | ALA5172262 | 24 | AUClast | = | 93.65 | ug/ml.min | ALA5144053 | ng.hr.mL-1 | ||||
16. | ALA5172262 | 24 | Tmax | = | 70 | min | ALA5144052 | hr | ||||
17. | ALA5172262 | 24 | Cmax | = | 0.301 | ug ml-1 | ALA5144051 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
18. | ALA5172262 | 24 | beta t1/2 | = | 289.9 | min | ALA5144050 | hr | ||||
19. | ALA5172262 | 24 | Drug metabolism | 0 | ALA5144049 | Metabolite_Detected | ||||||
20. | ALA5172262 | 24 | Drug metabolism | 0 | ALA5144048 | Metabolite_Detected |