| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5172456 | 8 | INH | 0 | ALA5130524 | NA | % | Homo sapiens | ||||
| 2. | ALA5172456 | 8 | F | = | 45 | % | ALA5130522 | % | ||||
| 3. | ALA5172456 | 8 | CL | = | 19 | ml/min.kg | ALA5130521 | mL.min-1.kg-1 | ||||
| 4. | ALA5172456 | 8 | F | = | 68 | % | ALA5130520 | % | ||||
| 5. | ALA5172456 | 8 | CL | = | 32 | ml/min.kg | ALA5130519 | mL.min-1.kg-1 | ||||
| 6. | ALA5172456 | 8 | IC50 | = | 19 | uM | ALA5130518 | 4.72 | nM | Homo sapiens | ||
| 7. | ALA5172456 | 8 | IC50 | > | 30 | uM | ALA5130517 | nM | Homo sapiens | |||
| 8. | ALA5172456 | 8 | IC50 | > | 30 | uM | ALA5130516 | nM | Homo sapiens | |||
| 9. | ALA5172456 | 8 | IC50 | > | 30 | uM | ALA5130515 | nM | Homo sapiens | |||
| 10. | ALA5172456 | 8 | IC50 | > | 40 | uM | ALA5130514 | nM | Homo sapiens | |||
| 11. | ALA5172456 | 8 | Papp | = | 6 | 10^-6 cm/s | ALA5130513 | 10^-6 cm/s | ||||
| 12. | ALA5172456 | 8 | CLH | = | 3.2 | uL/min | ALA5130512 | uL/min | ||||
| 13. | ALA5172456 | 8 | CLH | = | 3.2 | uL/min | ALA5130511 | uL/min | ||||
| 14. | ALA5172456 | 8 | CLH | < | 3 | uL/min | ALA5130510 | uL/min | ||||
| 15. | ALA5172456 | 8 | Therm_solubility | = | 42 | uM | ALA5130509 | nM | ||||
| 16. | ALA5172456 | 8 | logD | = | 1.2 | ALA5130508 | ||||||
| 17. | ALA5172456 | 8 | pKd | = | 5.4 | ALA5130507 | 5.40 | nM | Homo sapiens | |||
| 18. | ALA5172456 | 8 | FC | = | 0.78 | ALA5130504 | Homo sapiens | |||||
| 19. | ALA5172456 | 8 | Ratio IC50 | = | 87 | ALA5130503 | ||||||
| 20. | ALA5172456 | 8 | IC50 | = | 1.3 | uM | ALA5130502 | 5.89 | nM | Homo sapiens |
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