| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5172565 | 74 | EC50 | = | 119 | uM | ALA5158948 | nM | ||||
| 2. | ALA5172565 | 74 | Ratio | = | 0.93 | ALA5158947 | ||||||
| 3. | ALA5172565 | 74 | Papp | = | 3 | 10^-6 cm/s | ALA5158946 | 10^-6 cm/s | ||||
| 4. | ALA5172565 | 74 | Papp | = | 3.2 | 10^-6 cm/s | ALA5158945 | 10^-6 cm/s | ||||
| 5. | ALA5172565 | 74 | Ratio | = | 51.6 | ALA5158944 | ||||||
| 6. | ALA5172565 | 74 | Papp | = | 16.5 | 10^-6 cm/s | ALA5158943 | 10^-6 cm/s | ||||
| 7. | ALA5172565 | 74 | Papp | = | 0.32 | 10^-6 cm/s | ALA5158942 | 10^-6 cm/s | ||||
| 8. | ALA5172565 | 74 | log Pe | = | 5.03 | ALA5158941 | ||||||
| 9. | ALA5172565 | 74 | Drug recovery | = | 93 | % | ALA5158940 | % | ||||
| 10. | ALA5172565 | 74 | PPB | = | 85 | % | ALA5158939 | % | ||||
| 11. | ALA5172565 | 74 | CLH | = | 5.58 | uL/min | ALA5158938 | uL/min | ||||
| 12. | ALA5172565 | 74 | t1/2 | = | 251 | min | ALA5158937 | hr | ||||
| 13. | ALA5172565 | 74 | t1/2 | = | 568 | min | ALA5158936 | hr | ||||
| 14. | ALA5172565 | 74 | INH | 0 | ALA5158935 | NA | % | Homo sapiens | ||||
| 15. | ALA5172565 | 74 | INH | 0 | ALA5158934 | NA | % | Homo sapiens | ||||
| 16. | ALA5172565 | 74 | INH | 0 | ALA5158933 | NA | % | Homo sapiens | ||||
| 17. | ALA5172565 | 74 | INH | 0 | ALA5158932 | NA | % | Homo sapiens | ||||
| 18. | ALA5172565 | 74 | Kinact | = | 2.1 | /min | ALA5158930 | /min | Homo sapiens | |||
| 19. | ALA5172565 | 74 | Ki | = | 6.1 | uM | ALA5158930 | 5.21 | nM | Homo sapiens | ||
| 20. | ALA5172565 | 74 | Ratio | = | 352 | 10^3/M/min | ALA5158929 | 10^3/M/min | Homo sapiens |
The page will load shortly, Thanks for your patience!