# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5172581 | 7d | Activity | 0 | ALA5167241 | Non-Toxic | Homo sapiens | |||||
2. | ALA5172581 | 7d | solubility | = | 250 | ug ml-1 | ALA5167230 | ug.mL-1 | ||||
3. | ALA5172581 | 7d | Activity | 0 | ALA5167229 | Active | Homo sapiens | |||||
4. | ALA5172581 | 7d | Activity | 0 | ALA5167228 | Active | Mus musculus | |||||
5. | ALA5172581 | 7d | Activity | 0 | ALA5167227 | Active | Mus musculus | |||||
6. | ALA5172581 | 7d | Activity | 0 | ALA5167226 | Active | Mus musculus | |||||
7. | ALA5172581 | 7d | Activity | 0 | ALA5167225 | Active | Mus musculus | |||||
8. | ALA5172581 | 7d | Activity | 0 | ALA5167222 | Dde | Mus musculus | |||||
9. | ALA5172581 | 7d | FC | = | 1.71 | ALA5167221 | Mus musculus | |||||
10. | ALA5172581 | 7d | Kd | = | 0.429 | uM | ALA5167220 | 6.37 | nM | Homo sapiens | ||
11. | ALA5172581 | 7d | deltaTm | = | 3.3 | degrees C | ALA5167219 | degrees C | Homo sapiens | |||
12. | ALA5172581 | 7d | IC50 | = | 0.575 | uM | ALA5167218 | 6.24 | nM | Homo sapiens | ||
13. | ALA5172581 | 7d | Activity | 0 | ALA5167215 | Active | Mus musculus | |||||
14. | ALA5172581 | 7d | IC50 | = | 0.79 | uM | ALA5123054 | 6.10 | nM | Homo sapiens | ||
15. | ALA5172581 | 7d | INH | = | 56 | % | ALA5123053 | % | Homo sapiens | |||
16. | ALA5172581 | 7d | INH | = | 97 | % | ALA5123052 | % | Homo sapiens | |||
17. | ALA5172581 | 7d | INH | = | 96 | % | ALA5123051 | % | Homo sapiens |