# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5172913 | 6c | Ki | > | 4000 | nM | ALA5167425 | nM | Homo sapiens | |||
2. | ALA5172913 | 6c | Ki | > | 4000 | nM | ALA5167424 | nM | Homo sapiens | |||
3. | ALA5172913 | 6c | BPR | = | 0.32 | ALA5167423 | ||||||
4. | ALA5172913 | 6c | AUC | = | 69 | ng/mL.hr | ALA5167422 | ng.hr.mL-1 | ||||
5. | ALA5172913 | 6c | Cmax | = | 259 | ng/ml | ALA5167421 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
6. | ALA5172913 | 6c | Tmax | = | 0.17 | hr | ALA5167420 | hr | ||||
7. | ALA5172913 | 6c | t1/2 | = | 0.18 | hr | ALA5167419 | hr | ||||
8. | ALA5172913 | 6c | Kp | = | 0.29 | ALA5167418 | ||||||
9. | ALA5172913 | 6c | Ct | = | 23.6 | ng/g | ALA5167417 | ng/g | ||||
10. | ALA5172913 | 6c | Cp | = | 79.6 | ng/ml | ALA5167416 | ng/ml | ||||
11. | ALA5172913 | 6c | PPB | = | 2.2 | % | ALA5167415 | % | ||||
12. | ALA5172913 | 6c | PPB | = | 0.4 | % | ALA5167414 | % | ||||
13. | ALA5172913 | 6c | CLH | = | 1659 | ml/min.kg | ALA5167413 | mL.min-1.kg-1 | ||||
14. | ALA5172913 | 6c | CLH | = | 79.1 | ml/min.kg | ALA5167412 | mL.min-1.kg-1 | ||||
15. | ALA5172913 | 6c | EC50 | = | 0.014 | uM | ALA5167411 | 7.85 | nM | Homo sapiens | ||
16. | ALA5172913 | 6c | Emax | = | 82.2 | % | ALA5167410 | % | Homo sapiens | |||
17. | ALA5172913 | 6c | Ki | = | 271 | nM | ALA5167409 | 6.57 | nM | Homo sapiens | ||
18. | ALA5172913 | 6c | CL | = | 36.7 | ml/min.kg | ALA5167408 | mL.min-1.kg-1 | ||||
19. | ALA5172913 | 6c | t1/2 | = | 0.48 | hr | ALA5167407 | hr | ||||
20. | ALA5172913 | 6c | AUC | = | 119 | ng/mL.hr | ALA5167406 | ng.hr.mL-1 |