| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5175064 | 53 | Activity | 0 | ALA5132115 | NA | Mus musculus | |||||
| 2. | ALA5175064 | 53 | BPR | = | 0.34 | ALA5132113 | ||||||
| 3. | ALA5175064 | 53 | Cmax | = | 576 | ng/ml | ALA5132112 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 4. | ALA5175064 | 53 | CL | = | 21 | ml/min.kg | ALA5132111 | mL.min-1.kg-1 | ||||
| 5. | ALA5175064 | 53 | t1/2 | = | 5.6 | hr | ALA5132110 | hr | ||||
| 6. | ALA5175064 | 53 | Cmax | = | 1670 | ng/ml | ALA5132109 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 7. | ALA5175064 | 53 | Ratio | = | 1.8 | ALA5132108 | ||||||
| 8. | ALA5175064 | 53 | Papp | = | 23.5 | 10^-6 cm/s | ALA5132107 | 10^-6 cm/s | ||||
| 9. | ALA5175064 | 53 | Papp | = | 13.3 | 10^-6 cm/s | ALA5132106 | 10^-6 cm/s | ||||
| 10. | ALA5175064 | 53 | Ratio EC50 | = | 3 | ALA5132105 | Homo sapiens | |||||
| 11. | ALA5175064 | 53 | EC50 | = | 6.5 | uM | ALA5132104 | 5.19 | nM | Mus musculus | ||
| 12. | ALA5175064 | 53 | EC50 | = | 8.9 | uM | ALA5132103 | 5.05 | nM | Mus musculus | ||
| 13. | ALA5175064 | 53 | Emax | = | 270 | % | ALA5132102 | % | Mus musculus | |||
| 14. | ALA5175064 | 53 | Emax | = | 92 | % | ALA5132101 | % | Homo sapiens | |||
| 15. | ALA5175064 | 53 | pEC50 | = | 7.86 | ALA5132100 | 7.86 | nM | Homo sapiens | |||
| 16. | ALA5175064 | 53 | EC50 | = | 14 | nM | ALA5132100 | 7.85 | nM | Homo sapiens | ||
| 17. | ALA5175064 | 53 | Emax | = | 320 | % | ALA5132099 | % | Mus musculus |
The page will load shortly, Thanks for your patience!