# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5177715 | 15g | CL | = | 7.16 | ml/min.kg | ALA5148242 | mL.min-1.kg-1 | ||||
2. | ALA5177715 | 15g | Kp | = | 0.61 | ALA5148241 | ||||||
3. | ALA5177715 | 15g | Kp | = | 2.4 | ALA5148240 | ||||||
4. | ALA5177715 | 15g | Cmax | = | 68.7 | ng/ml | ALA5148239 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
5. | ALA5177715 | 15g | AUC | = | 288 | ng.hr/ml | ALA5148238 | ng.hr.mL-1 | ||||
6. | ALA5177715 | 15g | Stability | = | 91 | % | ALA5148237 | % | ||||
7. | ALA5177715 | 15g | Stability | > | 99 | % | ALA5148236 | % | ||||
8. | ALA5177715 | 15g | IC50 | > | 10 | uM | ALA5148235 | nM | Homo sapiens | |||
9. | ALA5177715 | 15g | IC50 | > | 10 | uM | ALA5148234 | nM | Homo sapiens | |||
10. | ALA5177715 | 15g | IC50 | > | 10 | uM | ALA5148233 | nM | Homo sapiens | |||
11. | ALA5177715 | 15g | IC50 | > | 10 | uM | ALA5148232 | nM | Homo sapiens | |||
12. | ALA5177715 | 15g | IC50 | > | 10 | uM | ALA5148231 | nM | Homo sapiens | |||
13. | ALA5177715 | 15g | Fu | = | 1.6 | % | ALA5148230 | |||||
14. | ALA5177715 | 15g | EC150 | = | 0.001 | uM | ALA5148229 | uM | Homo sapiens |