| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5178033 | 2b | INH | 0 | ALA5152891 | Active | % | |||||
| 2. | ALA5178033 | 2b | Ratio | = | 1.6 | ALA5152890 | ||||||
| 3. | ALA5178033 | 2b | Ratio | = | 7.8 | ALA5152889 | ||||||
| 4. | ALA5178033 | 2b | K(p,uu,brain) | = | 0.11 | ALA5152888 | ||||||
| 5. | ALA5178033 | 2b | Drug uptake(free) | = | 43 | nM | ALA5152887 | nM | ||||
| 6. | ALA5178033 | 2b | Cp(f) | = | 387 | nM | ALA5152886 | nM | ||||
| 7. | ALA5178033 | 2b | Ct | = | 1145 | ng/g | ALA5152885 | ng/g | ||||
| 8. | ALA5178033 | 2b | Cp | = | 1943 | ng/ml | ALA5152884 | ng/ml | ||||
| 9. | ALA5178033 | 2b | Fu | = | 0.017 | ALA5152883 | ||||||
| 10. | ALA5178033 | 2b | Fu | = | 0.09 | ALA5152882 | ||||||
| 11. | ALA5178033 | 2b | IC50 | = | 5.5 | nM | ALA5152881 | 8.26 | nM | Mus musculus | ||
| 12. | ALA5178033 | 2b | CLH | = | 4 | microL/min/mg | ALA5152880 | mL.min-1.g-1 | ||||
| 13. | ALA5178033 | 2b | CLH | = | -18 | microL/min/mg | ALA5152879 | mL.min-1.g-1 | ||||
| 14. | ALA5178033 | 2b | Kinetic_solubility | = | 1.9 | ug ml-1 | ALA5152878 | ug.mL-1 | ||||
| 15. | ALA5178033 | 2b | logD | = | 2.85 | ALA5152877 | ||||||
| 16. | ALA5178033 | 2b | Ratio | = | 4.5 | ALA5152876 | ||||||
| 17. | ALA5178033 | 2b | IC50 | = | 5.9 | nM | ALA5152875 | 8.23 | nM | Homo sapiens |
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