# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | CHR-6494 | 62; CHR-6494 | IC50 | = | 2 | nM | ALA5097328 | 8.70 | nM | Homo sapiens | ||
2. | CHR-6494 | 62; CHR-6494 | INH | 0 | ALA5165935 | Active | % | Homo sapiens | ||||
3. | CHR-6494 | 62; CHR-6494 | Selectivity Index | = | 2.7 | ALA5165921 | ||||||
4. | CHR-6494 | 62; CHR-6494 | IC50 | = | 119 | nM | ALA5165920 | 6.92 | nM | Homo sapiens | ||
5. | CHR-6494 | 62; CHR-6494 | Activity | = | 19 | % | ALA5165919 | % | Homo sapiens | |||
6. | CHR-6494 | 62; CHR-6494 | IC50 | = | 162 | nM | ALA5165918 | 6.79 | nM | Homo sapiens | ||
7. | CHR-6494 | 62; CHR-6494 | Activity | = | 13 | % | ALA5165917 | % | Homo sapiens | |||
8. | CHR-6494 | 62; CHR-6494 | Activity | = | 20 | % | ALA5165916 | % | Homo sapiens | |||
9. | CHR-6494 | 62; CHR-6494 | IC50 | = | 41 | nM | ALA5165915 | 7.39 | nM | Homo sapiens | ||
10. | CHR-6494 | 62; CHR-6494 | IC50 | = | 99 | nM | ALA5165914 | 7.00 | nM | Homo sapiens | ||
11. | CHR-6494 | 62; CHR-6494 | Activity | = | 6 | % | ALA5165913 | % | Homo sapiens | |||
12. | CHR-6494 | 62; CHR-6494 | IC50 | = | 53 | nM | ALA5165912 | 7.28 | nM | Homo sapiens | ||
13. | CHR-6494 | 62; CHR-6494 | Activity | = | 10 | % | ALA5165911 | % | Homo sapiens | |||
14. | CHR-6494 | 62; CHR-6494 | IC50 | = | 29 | nM | ALA5165910 | 7.54 | nM | |||
15. | CHR-6494 | 62; CHR-6494 | Activity | = | 12 | % | ALA5165909 | % | Homo sapiens | |||
16. | CHR-6494 | 62; CHR-6494 | IC50 | = | 13 | nM | ALA5165908 | 7.89 | nM | Rattus norvegicus | ||
17. | CHR-6494 | 62; CHR-6494 | Activity | = | 6 | % | ALA5165907 | % | Rattus norvegicus | |||
18. | CHR-6494 | 62; CHR-6494 | IC50 | = | 8 | nM | ALA5165906 | 8.10 | nM | Mus musculus | ||
19. | CHR-6494 | 62; CHR-6494 | Activity | = | 0 | % | ALA5165905 | % | Mus musculus | |||
20. | CHR-6494 | 62; CHR-6494 | IC50 | = | 3 | nM | ALA5165904 | 8.52 | nM | Homo sapiens |