# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5180080 | (R)-8i | F | = | 0.36 | % | ALA5156061 | % | ||||
2. | ALA5180080 | (R)-8i | t1/2 | = | 0.39 | hr | ALA5156060 | hr | ||||
3. | ALA5180080 | (R)-8i | Ct | = | 110.4 | nM | ALA5156059 | nM | ||||
4. | ALA5180080 | (R)-8i | Cp | = | 55.5 | nM | ALA5156058 | nM | ||||
5. | ALA5180080 | (R)-8i | Activity | 0 | ALA5156057 | Non-Toxic | ||||||
6. | ALA5180080 | (R)-8i | Activity | 0 | ALA5156056 | Non-Toxic | ||||||
7. | ALA5180080 | (R)-8i | Activity | 0 | ALA5156055 | Non-Toxic | ||||||
8. | ALA5180080 | (R)-8i | Activity | 0 | ALA5156054 | Non-Toxic | ||||||
9. | ALA5180080 | (R)-8i | Activity | 0 | ALA5156053 | Non-Toxic | ||||||
10. | ALA5180080 | (R)-8i | Activity | 0 | ALA5156052 | Non-Toxic | ||||||
11. | ALA5180080 | (R)-8i | Activity | 0 | ALA5156051 | Non-Toxic | ||||||
12. | ALA5180080 | (R)-8i | Activity | 0 | ALA5156050 | Non-Toxic | ||||||
13. | ALA5180080 | (R)-8i | Activity | 0 | ALA5156049 | Non-Toxic | ||||||
14. | ALA5180080 | (R)-8i | Activity | 0 | ALA5156048 | Active | Homo sapiens | |||||
15. | ALA5180080 | (R)-8i | Activity | 0 | ALA5156047 | Non-Toxic | ||||||
16. | ALA5180080 | (R)-8i | TGI | = | 52.9 | % | ALA5156045 | % | Homo sapiens | |||
17. | ALA5180080 | (R)-8i | INH | = | 60 | % | ALA5156044 | % | Homo sapiens | |||
18. | ALA5180080 | (R)-8i | INH | = | 50 | % | ALA5156043 | % | Homo sapiens | |||
19. | ALA5180080 | (R)-8i | Activity | = | 10.21 | % | ALA5156042 | % | Homo sapiens | |||
20. | ALA5180080 | (R)-8i | Activity | = | 30.1 | % | ALA5156041 | % | Homo sapiens |