| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5180330 | 21 | Activity | 0 | ALA5155980 | NA | Mus musculus | |||||
| 2. | ALA5180330 | 21 | Ki | = | 2.21 | nM | ALA5155979 | 8.66 | nM | Mus musculus | ||
| 3. | ALA5180330 | 21 | Ki | = | 7050 | nM | ALA5155978 | 5.15 | nM | Mus musculus | ||
| 4. | ALA5180330 | 21 | Activity | 0 | ALA5155977 | Active | Mus musculus | |||||
| 5. | ALA5180330 | 21 | t1/2 | = | 2 | min | ALA5155976 | hr | ||||
| 6. | ALA5180330 | 21 | t1/2 | = | 11.5 | min | ALA5155975 | hr | ||||
| 7. | ALA5180330 | 21 | t1/2 | = | 6.72 | min | ALA5155974 | hr | ||||
| 8. | ALA5180330 | 21 | Ratio | = | 46.6 | ALA5155973 | ||||||
| 9. | ALA5180330 | 21 | Papp | = | 0.44 | 10^-6 cm/s | ALA5155972 | 10^-6 cm/s | ||||
| 10. | ALA5180330 | 21 | Stability | = | 100 | % | ALA5155971 | % | ||||
| 11. | ALA5180330 | 21 | Stability | = | 100 | % | ALA5155970 | % | ||||
| 12. | ALA5180330 | 21 | Stability | = | 100 | % | ALA5155969 | % | ||||
| 13. | ALA5180330 | 21 | IC50 | = | 0.78 | uM | ALA5155968 | 6.11 | nM | Homo sapiens | ||
| 14. | ALA5180330 | 21 | IC50 | = | 17.7 | uM | ALA5155967 | 4.75 | nM | Homo sapiens | ||
| 15. | ALA5180330 | 21 | IC50 | = | 15.1 | uM | ALA5155966 | 4.82 | nM | Homo sapiens | ||
| 16. | ALA5180330 | 21 | IC50 | > | 30 | uM | ALA5155965 | nM | Homo sapiens | |||
| 17. | ALA5180330 | 21 | IC50 | = | 0.43 | uM | ALA5155964 | 6.37 | nM | Homo sapiens | ||
| 18. | ALA5180330 | 21 | Stability | = | 100 | % | ALA5155963 | % | ||||
| 19. | ALA5180330 | 21 | Stability | = | 100 | % | ALA5155962 | % | ||||
| 20. | ALA5180330 | 21 | Ki | = | 8.67 | nM | ALA5155957 | 8.06 | nM | Homo sapiens |
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