| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5180826 | 1 | Activity | 0 | ALA5162515 | NA | Homo sapiens | |||||
| 2. | ALA5180826 | 1 | Activity | 0 | ALA5162514 | NA | Homo sapiens | |||||
| 3. | ALA5180826 | 1 | Activity | = | 37.67 | % | ALA5162513 | % | Homo sapiens | |||
| 4. | ALA5180826 | 1 | Activity | 0 | ALA5162512 | Active | Rattus norvegicus | |||||
| 5. | ALA5180826 | 1 | Activity | 0 | ALA5162511 | Active | Rattus norvegicus | |||||
| 6. | ALA5180826 | 1 | Kd | = | 146 | uM | ALA5162509 | nM | Homo sapiens | |||
| 7. | ALA5180826 | 1 | Activity | 0 | ALA5162508 | NA | Homo sapiens | |||||
| 8. | ALA5180826 | 1 | Activity | 0 | ALA5162507 | NA | Homo sapiens | |||||
| 9. | ALA5180826 | 1 | Activity | 0 | ALA5162503 | Active | Rattus norvegicus | |||||
| 10. | ALA5180826 | 1 | Activity | 0 | ALA5162502 | Active | Rattus norvegicus | |||||
| 11. | ALA5180826 | 1 | F | = | 43.8 | % | ALA5162501 | % | ||||
| 12. | ALA5180826 | 1 | MRT | = | 1.33 | hr | ALA5162500 | hr | ||||
| 13. | ALA5180826 | 1 | AUC | = | 653 | ng.hr/ml | ALA5162499 | ng.hr.mL-1 | ||||
| 14. | ALA5180826 | 1 | t1/2 | = | 1.37 | hr | ALA5162498 | hr | ||||
| 15. | ALA5180826 | 1 | Tmax | = | 0.25 | hr | ALA5162497 | hr | ||||
| 16. | ALA5180826 | 1 | Cmax | = | 612 | ng/ml | ALA5162496 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 17. | ALA5180826 | 1 | MRT | = | 0.262 | hr | ALA5162495 | hr | ||||
| 18. | ALA5180826 | 1 | AUC | = | 448 | ng.hr/ml | ALA5162494 | ng.hr.mL-1 | ||||
| 19. | ALA5180826 | 1 | CL | = | 112 | ml/min.kg | ALA5162493 | mL.min-1.kg-1 | ||||
| 20. | ALA5180826 | 1 | Vdss | = | 1.75 | L/Kg | ALA5162492 | L.kg-1 |
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