# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5180977 | 50; JH106 | INH | = | 45.3 | % | ALA5216332 | % | Homo sapiens | |||
2. | ALA5180977 | 50; JH106 | INH | = | 95.2 | % | ALA5216331 | % | Homo sapiens | |||
3. | ALA5180977 | 50; JH106 | IC50 | = | 6.4 | uM | ALA5216330 | 5.19 | nM | Homo sapiens | ||
4. | ALA5180977 | 50; JH106 | IC50 | = | 18 | uM | ALA5216329 | 4.75 | nM | Homo sapiens | ||
5. | ALA5180977 | 50; JH106 | IC50 | = | 5.9 | uM | ALA5216328 | 5.23 | nM | Homo sapiens | ||
6. | ALA5180977 | 50; JH106 | IC50 | = | 3.7 | uM | ALA5216327 | 5.43 | nM | Homo sapiens | ||
7. | ALA5180977 | 50; JH106 | INH | 0 | ALA5135141 | Active | % | Homo sapiens | ||||
8. | ALA5180977 | 50; JH106 | INH | 0 | ALA5135140 | Dde | % | Homo sapiens | ||||
9. | ALA5180977 | 50; JH106 | INH | = | 42 | % | ALA5135139 | % | Homo sapiens | |||
10. | ALA5180977 | 50; JH106 | INH | 0 | ALA5135138 | Tde | % | Homo sapiens | ||||
11. | ALA5180977 | 50; JH106 | INH | 0 | ALA5135138 | Dde | % | Homo sapiens | ||||
12. | ALA5180977 | 50; JH106 | FC | > | 1.5 | ALA5135128 | Homo sapiens | |||||
13. | ALA5180977 | 50; JH106 | IC50 | = | 6.4 | uM | ALA5135127 | 5.19 | nM | Homo sapiens | ||
14. | ALA5180977 | 50; JH106 | IC50 | = | 18 | uM | ALA5135126 | 4.75 | nM | Homo sapiens | ||
15. | ALA5180977 | 50; JH106 | IC50 | = | 5.9 | uM | ALA5135125 | 5.23 | nM | Homo sapiens | ||
16. | ALA5180977 | 50; JH106 | IC50 | = | 3.7 | uM | ALA5135124 | 5.43 | nM | Homo sapiens | ||
17. | ALA5180977 | 50; JH106 | INH | = | 45.3 | % | ALA5135119 | % | Homo sapiens | |||
18. | ALA5180977 | 50; JH106 | INH | = | 95.2 | % | ALA5135116 | % | Homo sapiens | |||
19. | ALA5180977 | 50; JH106 | deltaTm | = | 1.4 | degrees C | ALA5135115 | degrees C |