# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | D6808 | 14; D6808 | IC50 | = | 27.72 | uM | ALA5100299 | 4.56 | nM | Homo sapiens | ||
2. | D6808 | 14; D6808 | IC50 | > | 10 | uM | ALA5100298 | nM | Homo sapiens | |||
3. | D6808 | 14; D6808 | IC50 | > | 10 | uM | ALA5100297 | nM | Homo sapiens | |||
4. | D6808 | 14; D6808 | IC50 | > | 10 | uM | ALA5100296 | nM | Homo sapiens | |||
5. | D6808 | 14; D6808 | F | = | 33.91 | % | ALA5100295 | % | ||||
6. | D6808 | 14; D6808 | F | = | 2.02 | % | ALA5100294 | % | ||||
7. | D6808 | 14; D6808 | MRT(t) | = | 3.4 | hr | ALA5100293 | hr | ||||
8. | D6808 | 14; D6808 | MRT(t) | = | 1.71 | hr | ALA5100292 | hr | ||||
9. | D6808 | 14; D6808 | MRT(t) | = | 0.36 | hr | ALA5100291 | hr | ||||
10. | D6808 | 14; D6808 | CL | = | 4207.06 | ml/hr/kg | ALA5100290 | mL.min-1.kg-1 | ||||
11. | D6808 | 14; D6808 | Vz | = | 3470.78 | ml/kg | ALA5100289 | L.kg-1 | ||||
12. | D6808 | 14; D6808 | Cmax | = | 282.12 | ng/ml | ALA5100288 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
13. | D6808 | 14; D6808 | Cmax | = | 60.98 | ng/ml | ALA5100287 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
14. | D6808 | 14; D6808 | Cmax | = | 1071.23 | ng/ml | ALA5100286 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
15. | D6808 | 14; D6808 | Tmax | = | 0.25 | hr | ALA5100285 | hr | ||||
16. | D6808 | 14; D6808 | Tmax | = | 0.25 | hr | ALA5100284 | hr | ||||
17. | D6808 | 14; D6808 | Tmax | = | 0.08 | hr | ALA5100283 | hr | ||||
18. | D6808 | 14; D6808 | t1/2 | = | 4.63 | hr | ALA5100282 | hr | ||||
19. | D6808 | 14; D6808 | t1/2 | = | 2.49 | hr | ALA5100281 | hr | ||||
20. | D6808 | 14; D6808 | t1/2 | = | 0.57 | hr | ALA5100280 | hr |