| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5181694 | 19 | F | = | 13.71 | % | ALA5162333 | % | ||||
| 2. | ALA5181694 | 19 | t1/2 | = | 4.14 | hr | ALA5162332 | hr | ||||
| 3. | ALA5181694 | 19 | AUCt | = | 0.17 | hr.microg/ml | ALA5162331 | ng.hr.mL-1 | ||||
| 4. | ALA5181694 | 19 | Tmax | = | 2.67 | hr | ALA5162330 | hr | ||||
| 5. | ALA5181694 | 19 | Cmax | = | 0.03 | ug ml-1 | ALA5162329 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 6. | ALA5181694 | 19 | Vdss | = | 23.64 | L/Kg | ALA5162328 | L.kg-1 | ||||
| 7. | ALA5181694 | 19 | t1/2 | = | 6.62 | hr | ALA5162327 | hr | ||||
| 8. | ALA5181694 | 19 | F | = | 34.43 | % | ALA5162325 | % | ||||
| 9. | ALA5181694 | 19 | t1/2 | = | 0.87 | hr | ALA5162324 | hr | ||||
| 10. | ALA5181694 | 19 | AUCt | = | 0.63 | hr.microg/ml | ALA5162323 | ng.hr.mL-1 | ||||
| 11. | ALA5181694 | 19 | Tmax | = | 0.42 | hr | ALA5162322 | hr | ||||
| 12. | ALA5181694 | 19 | Cmax | = | 0.29 | ug ml-1 | ALA5162321 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 13. | ALA5181694 | 19 | Vdss | = | 4.49 | L/Kg | ALA5162320 | L.kg-1 | ||||
| 14. | ALA5181694 | 19 | t1/2 | = | 1.16 | hr | ALA5162319 | hr | ||||
| 15. | ALA5181694 | 19 | CL | = | 4.85 | L/Kg.hr | ALA5162317 | L/Kg.hr | ||||
| 16. | ALA5181694 | 19 | CL | = | 5.4 | L/Kg.hr | ALA5162316 | L/Kg.hr | ||||
| 17. | ALA5181694 | 19 | CLH | = | 11.77 | microL/min/mg | ALA5162315 | mL.min-1.g-1 | ||||
| 18. | ALA5181694 | 19 | t1/2 | = | 117.77 | min | ALA5162314 | hr | ||||
| 19. | ALA5181694 | 19 | Ratio IC50 | = | 64.1 | ALA5162312 | Homo sapiens | |||||
| 20. | ALA5181694 | 19 | Ratio IC50 | = | 70.5 | ALA5162311 | Homo sapiens |
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