# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5181908 | 7q | Ratio IC50 | > | 100 | ALA5161312 | ||||||
2. | ALA5181908 | 7q | Ratio IC50 | = | 3 | ALA5161311 | Homo sapiens | |||||
3. | ALA5181908 | 7q | Kel | = | 1.133 | /hr | ALA5161309 | /hr | ||||
4. | ALA5181908 | 7q | Kel | = | 12.076 | /hr | ALA5161308 | /hr | ||||
5. | ALA5181908 | 7q | ka | = | 1.65 | /hr | ALA5161307 | /hr | ||||
6. | ALA5181908 | 7q | IC50 | = | 7.45 | uM | ALA5161306 | 5.13 | nM | Homo sapiens | ||
7. | ALA5181908 | 7q | IC50 | > | 100 | uM | ALA5161305 | nM | Homo sapiens | |||
8. | ALA5181908 | 7q | IC50 | > | 100 | uM | ALA5161304 | nM | Homo sapiens | |||
9. | ALA5181908 | 7q | solubility | = | 26 | ug ml-1 | ALA5161303 | ug.mL-1 | ||||
10. | ALA5181908 | 7q | BPR | = | 1.66 | ALA5161302 | ||||||
11. | ALA5181908 | 7q | Cp | = | 1405 | ng/g | ALA5161301 | ng/g | ||||
12. | ALA5181908 | 7q | Ct | = | 2311 | ng/g | ALA5161300 | ng/g | ||||
13. | ALA5181908 | 7q | F | = | 60 | % | ALA5161299 | % | ||||
14. | ALA5181908 | 7q | MRT | = | 1.426 | hr | ALA5161298 | hr | ||||
15. | ALA5181908 | 7q | MRT | = | 0.153 | hr | ALA5161297 | hr | ||||
16. | ALA5181908 | 7q | AUC | = | 598.873 | ng/mL.hr | ALA5161296 | ng.hr.mL-1 | ||||
17. | ALA5181908 | 7q | AUC | = | 495.955 | ng/mL.hr | ALA5161295 | ng.hr.mL-1 | ||||
18. | ALA5181908 | 7q | CL | = | 0.022 | L/hr/kg | ALA5161294 | mL.min-1.kg-1 | ||||
19. | ALA5181908 | 7q | CL | = | 0.024 | L/hr/kg | ALA5161293 | mL.min-1.kg-1 | ||||
20. | ALA5181908 | 7q | Cmax | = | 311.377 | ng/ml | ALA5161292 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM |