# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5183586 | 7 | Drug uptake | = | 5.4 | % | ALA5159125 | % | ||||
2. | ALA5183586 | 7 | deltaTm | = | 1 | degrees C | ALA5159120 | degrees C | Homo sapiens | |||
3. | ALA5183586 | 7 | Selectivity Index | = | 69.3 | ALA5159119 | ||||||
4. | ALA5183586 | 7 | Selectivity Index | = | 1.3 | ALA5159118 | ||||||
5. | ALA5183586 | 7 | Selectivity Index | = | 2.9 | ALA5159117 | ||||||
6. | ALA5183586 | 7 | IC50 | = | 10.4 | uM | ALA5159116 | 4.98 | nM | Homo sapiens | ||
7. | ALA5183586 | 7 | IC50 | = | 3.6 | uM | ALA5159115 | 5.44 | nM | Homo sapiens | ||
8. | ALA5183586 | 7 | IC50 | = | 27.5 | uM | ALA5159114 | 4.56 | nM | Leishmania major | ||
9. | ALA5183586 | 7 | IC50 | = | 0.15 | uM | ALA5159113 | 6.82 | nM | Trypanosoma brucei | ||
10. | ALA5183586 | 7 | deltaTm | = | 5 | degrees C | ALA5159128 | degrees C | Homo sapiens |