# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5184610 | 14 | INH | 0 | ALA5162371 | NA | % | Homo sapiens | ||||
2. | ALA5184610 | 14 | F | = | 47.48 | % | ALA5162333 | % | ||||
3. | ALA5184610 | 14 | t1/2 | = | 4.32 | hr | ALA5162332 | hr | ||||
4. | ALA5184610 | 14 | AUCt | = | 2.17 | hr.microg/ml | ALA5162331 | ng.hr.mL-1 | ||||
5. | ALA5184610 | 14 | Tmax | = | 4 | hr | ALA5162330 | hr | ||||
6. | ALA5184610 | 14 | Cmax | = | 0.28 | ug ml-1 | ALA5162329 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
7. | ALA5184610 | 14 | Vdss | = | 10.6 | L/Kg | ALA5162328 | L.kg-1 | ||||
8. | ALA5184610 | 14 | t1/2 | = | 2.09 | hr | ALA5162327 | hr | ||||
9. | ALA5184610 | 14 | F | = | 22.6 | % | ALA5162325 | % | ||||
10. | ALA5184610 | 14 | t1/2 | = | 3.07 | hr | ALA5162324 | hr | ||||
11. | ALA5184610 | 14 | AUCt | = | 1.7 | hr.microg/ml | ALA5162323 | ng.hr.mL-1 | ||||
12. | ALA5184610 | 14 | Tmax | = | 1.67 | hr | ALA5162322 | hr | ||||
13. | ALA5184610 | 14 | Cmax | = | 0.4 | ug ml-1 | ALA5162321 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
14. | ALA5184610 | 14 | Vdss | = | 2.79 | L/Kg | ALA5162320 | L.kg-1 | ||||
15. | ALA5184610 | 14 | t1/2 | = | 4.38 | hr | ALA5162319 | hr | ||||
16. | ALA5184610 | 14 | CL | = | 3.33 | L/Kg.hr | ALA5162317 | L/Kg.hr | ||||
17. | ALA5184610 | 14 | CL | = | 1.32 | L/Kg.hr | ALA5162316 | L/Kg.hr | ||||
18. | ALA5184610 | 14 | CLH | = | 1.81 | microL/min/mg | ALA5162315 | mL.min-1.g-1 | ||||
19. | ALA5184610 | 14 | t1/2 | = | 776.84 | min | ALA5162314 | hr | ||||
20. | ALA5184610 | 14 | Ratio IC50 | = | 7.4 | ALA5162312 | Homo sapiens |