| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5184829 | 7aa | Ratio IC50 | = | 81 | ALA5130182 | ||||||
| 2. | ALA5184829 | 7aa | IC50 | = | 25 | nM | ALA5130181 | 7.60 | nM | Rattus norvegicus | ||
| 3. | ALA5184829 | 7aa | Activity | = | 249 | ng/L | ALA5130180 | ng/L | ||||
| 4. | ALA5184829 | 7aa | Activity | = | 28 | ng/L | ALA5130179 | ng/L | ||||
| 5. | ALA5184829 | 7aa | F | = | 21.4 | % | ALA5130178 | % | ||||
| 6. | ALA5184829 | 7aa | CL | = | 17.2 | ml/hr/kg | ALA5130177 | mL.min-1.kg-1 | ||||
| 7. | ALA5184829 | 7aa | beta t1/2 | = | 4.6 | hr | ALA5130176 | hr | ||||
| 8. | ALA5184829 | 7aa | beta t1/2 | = | 4.5 | hr | ALA5130175 | hr | ||||
| 9. | ALA5184829 | 7aa | AUC | = | 54539.2 | ug/L.hr | ALA5130174 | ng.hr.mL-1 | ||||
| 10. | ALA5184829 | 7aa | AUC | = | 50928.7 | ug/L.hr | ALA5130173 | ng.hr.mL-1 | ||||
| 11. | ALA5184829 | 7aa | Tmax | = | 4.2 | hr | ALA5130172 | hr | ||||
| 12. | ALA5184829 | 7aa | Tmax | = | 0 | hr | ALA5130171 | hr | ||||
| 13. | ALA5184829 | 7aa | Cmax | = | 7993.3 | ug/L | ALA5130170 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 14. | ALA5184829 | 7aa | Cmax | = | 12685.7 | ug/L | ALA5130169 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 15. | ALA5184829 | 7aa | LC50 | > | 50 | uM | ALA5130168 | nM | Cricetulus griseus | |||
| 16. | ALA5184829 | 7aa | LC50 | > | 50 | uM | ALA5130167 | nM | Homo sapiens | |||
| 17. | ALA5184829 | 7aa | solubility | = | 196 | uM | ALA5130166 | nM | ||||
| 18. | ALA5184829 | 7aa | IC50 | > | 10 | uM | ALA5130165 | nM | Homo sapiens | |||
| 19. | ALA5184829 | 7aa | IC50 | > | 10 | uM | ALA5130164 | nM | Homo sapiens | |||
| 20. | ALA5184829 | 7aa | IC50 | > | 10 | uM | ALA5130163 | nM | Homo sapiens |
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