# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5185902 | 39 | F | = | 23 | % | ALA5139001 | % | ||||
2. | ALA5185902 | 39 | AUC | = | 708 | nM.hr | ALA5139000 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
3. | ALA5185902 | 39 | t1/2 | = | 5.2 | hr | ALA5138999 | hr | ||||
4. | ALA5185902 | 39 | Vdss | = | 3.9 | L/Kg | ALA5138998 | L.kg-1 | ||||
5. | ALA5185902 | 39 | CL | = | 54 | ml/min.kg | ALA5138997 | mL.min-1.kg-1 | ||||
6. | ALA5185902 | 39 | ERH | = | 78 | % | ALA5138996 | % | ||||
7. | ALA5185902 | 39 | ERH | = | 49 | % | ALA5138995 | % | ||||
8. | ALA5185902 | 39 | IC50 | = | 37 | nM | ALA5138981 | 7.43 | nM | |||
9. | ALA5185902 | 39 | IC50 | = | 147 | nM | ALA5138980 | 6.83 | nM | Rattus norvegicus | ||
10. | ALA5185902 | 39 | IC50 | = | 94 | nM | ALA5138979 | 7.03 | nM | Rattus norvegicus | ||
11. | ALA5185902 | 39 | IC50 | = | 2577 | nM | ALA5138978 | 5.59 | nM | Homo sapiens |