# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5186093 | 6 | INH | 0 | ALA5165935 | Active | % | Homo sapiens | ||||
2. | ALA5186093 | 6 | Activity | 0 | ALA5165933 | Dde | Homo sapiens | |||||
3. | ALA5186093 | 6 | Activity | 0 | ALA5165932 | Dde | Homo sapiens | |||||
4. | ALA5186093 | 6 | EC50 | = | 0.2 | uM | ALA5165926 | 6.70 | nM | Homo sapiens | ||
5. | ALA5186093 | 6 | EC50 | = | 0.8 | uM | ALA5165925 | 6.10 | nM | Homo sapiens | ||
6. | ALA5186093 | 6 | EC50 | = | 0.2 | uM | ALA5165924 | 6.70 | nM | Homo sapiens | ||
7. | ALA5186093 | 6 | EC50 | = | 0.4 | uM | ALA5165923 | 6.40 | nM | Homo sapiens | ||
8. | ALA5186093 | 6 | EC50 | = | 0.3 | uM | ALA5165922 | 6.52 | nM | Homo sapiens | ||
9. | ALA5186093 | 6 | Selectivity Index | = | 6.7 | ALA5165921 | ||||||
10. | ALA5186093 | 6 | Activity | = | 42 | % | ALA5165919 | % | Homo sapiens | |||
11. | ALA5186093 | 6 | Activity | = | 94 | % | ALA5165917 | % | Homo sapiens | |||
12. | ALA5186093 | 6 | Activity | = | 91 | % | ALA5165916 | % | Homo sapiens | |||
13. | ALA5186093 | 6 | Activity | = | 55 | % | ALA5165913 | % | Homo sapiens | |||
14. | ALA5186093 | 6 | IC50 | = | 418 | nM | ALA5165912 | 6.38 | nM | Homo sapiens | ||
15. | ALA5186093 | 6 | Activity | = | 29 | % | ALA5165911 | % | Homo sapiens | |||
16. | ALA5186093 | 6 | IC50 | = | 24 | nM | ALA5165910 | 7.62 | nM | |||
17. | ALA5186093 | 6 | Activity | = | 9 | % | ALA5165909 | % | Homo sapiens | |||
18. | ALA5186093 | 6 | IC50 | = | 87 | nM | ALA5165908 | 7.06 | nM | Rattus norvegicus | ||
19. | ALA5186093 | 6 | Activity | = | 15 | % | ALA5165907 | % | Rattus norvegicus | |||
20. | ALA5186093 | 6 | IC50 | = | 20 | nM | ALA5165906 | 7.70 | nM | Mus musculus |