# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5186617 | 12e; EML979 | Time | = | 66.7 | s | ALA5138966 | hr | Homo sapiens | |||
2. | ALA5186617 | 12e; EML979 | K | = | 0.015 | 1/s | ALA5138965 | 1/s | Homo sapiens | |||
3. | ALA5186617 | 12e; EML979 | K | = | 2.58 | 10^4/Ms | ALA5138964 | 10^4/Ms | Homo sapiens | |||
4. | ALA5186617 | 12e; EML979 | Kd | = | 603.4 | nM | ALA5138963 | 6.22 | nM | Homo sapiens | ||
5. | ALA5186617 | 12e; EML979 | Selectivity Index | = | 33 | ALA5138956 | ||||||
6. | ALA5186617 | 12e; EML979 | Selectivity Index | = | 4 | ALA5138955 | ||||||
7. | ALA5186617 | 12e; EML979 | Selectivity Index | = | 202 | ALA5138954 | ||||||
8. | ALA5186617 | 12e; EML979 | Selectivity Index | = | 19 | ALA5138953 | ||||||
9. | ALA5186617 | 12e; EML979 | Selectivity Index | = | 70 | ALA5138952 | ||||||
10. | ALA5186617 | 12e; EML979 | Selectivity Index | = | 15 | ALA5138951 | ||||||
11. | ALA5186617 | 12e; EML979 | IC50 | = | 5.84 | uM | ALA5138950 | 5.23 | nM | Homo sapiens | ||
12. | ALA5186617 | 12e; EML979 | IC50 | = | 0.631 | uM | ALA5138949 | 6.20 | nM | Homo sapiens | ||
13. | ALA5186617 | 12e; EML979 | IC50 | = | 35.6 | uM | ALA5138948 | 4.45 | nM | Homo sapiens | ||
14. | ALA5186617 | 12e; EML979 | IC50 | = | 3.38 | uM | ALA5138947 | 5.47 | nM | Homo sapiens | ||
15. | ALA5186617 | 12e; EML979 | IC50 | = | 0.176 | uM | ALA5138946 | 6.75 | nM | Homo sapiens | ||
16. | ALA5186617 | 12e; EML979 | IC50 | = | 12.4 | uM | ALA5138945 | 4.91 | nM | Homo sapiens | ||
17. | ALA5186617 | 12e; EML979 | IC50 | = | 2.6 | uM | ALA5138944 | 5.58 | nM | Homo sapiens |