| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5187422 | RP-6685 | AUC | = | 14.7 | uM.hr | ALA5111566 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 2. | ALA5187422 | RP-6685 | AUC | = | 32.6 | uM.hr | ALA5111565 | standard_value was converted from uM.hr to ng.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | standard_value was converted from uM.hr to ug.hr.mL-1 using the parent compound MW | ng.hr.mL-1 | |||
| 3. | ALA5187422 | RP-6685 | Activity | 0 | ALA5111564 | Active | Homo sapiens | |||||
| 4. | ALA5187422 | RP-6685 | Activity | 0 | ALA5111563 | Active | Homo sapiens | |||||
| 5. | ALA5187422 | RP-6685 | Activity | 0 | ALA5111561 | Non-Toxic | ||||||
| 6. | ALA5187422 | RP-6685 | Activity | 0 | ALA5111560 | Non-Toxic | ||||||
| 7. | ALA5187422 | RP-6685 | Activity | 0 | ALA5111559 | Non-Toxic | ||||||
| 8. | ALA5187422 | RP-6685 | Activity | 0 | ALA5111558 | Non-Toxic | ||||||
| 9. | ALA5187422 | RP-6685 | Activity | 0 | ALA5111557 | Active | Homo sapiens | |||||
| 10. | ALA5187422 | RP-6685 | Activity | 0 | ALA5111556 | NA | Homo sapiens | |||||
| 11. | ALA5187422 | RP-6685 | Activity | 0 | ALA5111555 | Active | Homo sapiens | |||||
| 12. | ALA5187422 | RP-6685 | IC50 | = | 2.147 | 10^-6M | ALA5111552 | 5.67 | nM | |||
| 13. | ALA5187422 | RP-6685 | F | = | 66 | % | ALA5111551 | % | ||||
| 14. | ALA5187422 | RP-6685 | t1/2 | = | 0.4 | hr | ALA5111550 | hr | ||||
| 15. | ALA5187422 | RP-6685 | Vdss | = | 1.1 | L/Kg | ALA5111549 | L.kg-1 | ||||
| 16. | ALA5187422 | RP-6685 | CL | = | 36.8 | ml/min.kg | ALA5111548 | mL.min-1.kg-1 | ||||
| 17. | ALA5187422 | RP-6685 | Ratio | = | 1.4 | ALA5111547 | ||||||
| 18. | ALA5187422 | RP-6685 | logPapp | = | 6.2 | ALA5111546 | ||||||
| 19. | ALA5187422 | RP-6685 | f(Cave) | = | 0.107 | uM | ALA5111545 | uM | ||||
| 20. | ALA5187422 | RP-6685 | IC50 | > | 15 | uM | ALA5111544 | nM | Homo sapiens |
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