# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5188431 | 15i | CL | = | 17 | ml/min.kg | ALA5148242 | mL.min-1.kg-1 | ||||
2. | ALA5188431 | 15i | Kp | = | 0.98 | ALA5148241 | ||||||
3. | ALA5188431 | 15i | Kp | = | 2.19 | ALA5148240 | ||||||
4. | ALA5188431 | 15i | Cmax | = | 44.8 | ng/ml | ALA5148239 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
5. | ALA5188431 | 15i | AUC | = | 111 | ng.hr/ml | ALA5148238 | ng.hr.mL-1 | ||||
6. | ALA5188431 | 15i | Stability | = | 83 | % | ALA5148237 | % | ||||
7. | ALA5188431 | 15i | Stability | > | 99 | % | ALA5148236 | % | ||||
8. | ALA5188431 | 15i | IC50 | > | 10 | uM | ALA5148235 | nM | Homo sapiens | |||
9. | ALA5188431 | 15i | IC50 | > | 10 | uM | ALA5148234 | nM | Homo sapiens | |||
10. | ALA5188431 | 15i | IC50 | > | 10 | uM | ALA5148233 | nM | Homo sapiens | |||
11. | ALA5188431 | 15i | IC50 | > | 10 | uM | ALA5148232 | nM | Homo sapiens | |||
12. | ALA5188431 | 15i | IC50 | > | 10 | uM | ALA5148231 | nM | Homo sapiens | |||
13. | ALA5188431 | 15i | Fu | = | 7.2 | % | ALA5148230 | |||||
14. | ALA5188431 | 15i | EC150 | = | 0.003 | uM | ALA5148229 | uM | Homo sapiens |