# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5191280 | 27; LDT540A | deltaTm | = | 6.8 | degrees C | ALA5158252 | degrees C | Homo sapiens | |||
2. | ALA5191280 | 27; LDT540A | deltaTm | = | 5.6 | degrees C | ALA5158251 | degrees C | Homo sapiens | |||
3. | ALA5191280 | 27; LDT540A | deltaTm | = | 3.8 | degrees C | ALA5158250 | degrees C | Homo sapiens | |||
4. | ALA5191280 | 27; LDT540A | Activity | 0 | ALA5158249 | Active | ||||||
5. | ALA5191280 | 27; LDT540A | Activity | 0 | ALA5158225 | Active | Mus musculus | |||||
6. | ALA5191280 | 27; LDT540A | Activity | 0 | ALA5158224 | Active | Mus musculus | |||||
7. | ALA5191280 | 27; LDT540A | Emax | = | 5 | % | ALA5158221 | % | Homo sapiens | |||
8. | ALA5191280 | 27; LDT540A | Emax | >= | 90 | % | ALA5158220 | % | Homo sapiens | |||
9. | ALA5191280 | 27; LDT540A | Emax | >= | 90 | % | ALA5158219 | % | Homo sapiens | |||
10. | ALA5191280 | 27; LDT540A | Emax | = | 21 | uM | ALA5158218 | uM | Homo sapiens | |||
11. | ALA5191280 | 27; LDT540A | EC50 | = | 1.78 | uM | ALA5158217 | 5.75 | nM | Homo sapiens | ||
12. | ALA5191280 | 27; LDT540A | EC50 | = | 0.7 | uM | ALA5158216 | 6.16 | nM | Homo sapiens | ||
13. | ALA5191280 | 27; LDT540A | Activity | 0 | ALA5158211 | Active | Mus musculus | |||||
14. | ALA5191280 | 27; LDT540A | Activity | 0 | ALA5158210 | Active | Homo sapiens | |||||
15. | ALA5191280 | 27; LDT540A | Activity | 0 | ALA5158209 | Active | Homo sapiens | |||||
16. | ALA5191280 | 27; LDT540A | Activity | 0 | ALA5158208 | Active | Homo sapiens | |||||
17. | ALA5191280 | 27; LDT540A | Stability | = | 90 | % | ALA5158207 | % | ||||
18. | ALA5191280 | 27; LDT540A | t1/2 | = | 835 | min | ALA5158206 | hr |