# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5191531 | 17 | Activity | 0 | ALA5162515 | NA | Homo sapiens | |||||
2. | ALA5191531 | 17 | Activity | 0 | ALA5162514 | NA | Homo sapiens | |||||
3. | ALA5191531 | 17 | Activity | = | 31.43 | % | ALA5162513 | % | Homo sapiens | |||
4. | ALA5191531 | 17 | Kd | = | 95.7 | uM | ALA5162509 | 4.02 | nM | Homo sapiens | ||
5. | ALA5191531 | 17 | Activity | 0 | ALA5162508 | NA | Homo sapiens | |||||
6. | ALA5191531 | 17 | Activity | 0 | ALA5162507 | NA | Homo sapiens | |||||
7. | ALA5191531 | 17 | IC50 | = | 37.8 | uM | ALA5162485 | 4.42 | nM | Homo sapiens | ||
8. | ALA5191531 | 17 | PPB | = | 99.5 | % | ALA5162484 | % | ||||
9. | ALA5191531 | 17 | t1/2 | > | 60 | min | ALA5162483 | hr | ||||
10. | ALA5191531 | 17 | IC50 | = | 4.96 | uM | ALA5162482 | 5.30 | nM | Homo sapiens | ||
11. | ALA5191531 | 17 | t1/2 | > | 216.8 | min | ALA5162481 | hr | ||||
12. | ALA5191531 | 17 | Papp | > | 0.023 | 10^-6 cm/s | ALA5162480 | 10^-6 cm/s | ||||
13. | ALA5191531 | 17 | EC50 | = | 2.64 | uM | ALA5162479 | 5.58 | nM | Mus musculus | ||
14. | ALA5191531 | 17 | EC50 | = | 1.16 | uM | ALA5162478 | 5.94 | nM | Mus musculus | ||
15. | ALA5191531 | 17 | EC50 | = | 1.43 | uM | ALA5162477 | 5.84 | nM | Rattus norvegicus | ||
16. | ALA5191531 | 17 | EC50 | = | 0.97 | uM | ALA5162476 | 6.01 | nM | Rattus norvegicus | ||
17. | ALA5191531 | 17 | solubility | > | 122.52 | mg/ml | ALA5162473 | ug.mL-1 | ||||
18. | ALA5191531 | 17 | CLH | < | 0.64 | uL/min | ALA5162472 | uL/min | ||||
19. | ALA5191531 | 17 | EC50 | = | 0.47 | uM | ALA5162471 | 6.33 | nM | Rattus norvegicus |