# | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
---|---|---|---|---|---|---|---|---|---|---|---|---|
1. | ALA5191769 | 12g; EML982 | Activity | = | 80 | % | ALA5138969 | % | Homo sapiens | |||
2. | ALA5191769 | 12g; EML982 | Activity | 0 | ALA5138968 | Non-Toxic | Homo sapiens | |||||
3. | ALA5191769 | 12g; EML982 | permeability | 0 | ALA5138967 | Impermeable | ||||||
4. | ALA5191769 | 12g; EML982 | Time | = | 76.9 | s | ALA5138966 | hr | Homo sapiens | |||
5. | ALA5191769 | 12g; EML982 | K | = | 0.013 | 1/s | ALA5138965 | 1/s | Homo sapiens | |||
6. | ALA5191769 | 12g; EML982 | K | = | 0.25 | 10^6/Ms | ALA5138964 | 10^6/Ms | Homo sapiens | |||
7. | ALA5191769 | 12g; EML982 | Kd | = | 51.7 | nM | ALA5138963 | 7.29 | nM | Homo sapiens | ||
8. | ALA5191769 | 12g; EML982 | Selectivity Index | = | 168 | ALA5138956 | ||||||
9. | ALA5191769 | 12g; EML982 | Selectivity Index | = | 557 | ALA5138955 | ||||||
10. | ALA5191769 | 12g; EML982 | Selectivity Index | = | 517 | ALA5138954 | ||||||
11. | ALA5191769 | 12g; EML982 | Selectivity Index | = | 93 | ALA5138953 | ||||||
12. | ALA5191769 | 12g; EML982 | Selectivity Index | = | 1583 | ALA5138952 | ||||||
13. | ALA5191769 | 12g; EML982 | Selectivity Index | = | 214 | ALA5138951 | ||||||
14. | ALA5191769 | 12g; EML982 | IC50 | = | 1.41 | uM | ALA5138950 | 5.85 | nM | Homo sapiens | ||
15. | ALA5191769 | 12g; EML982 | IC50 | = | 4.68 | uM | ALA5138949 | 5.33 | nM | Homo sapiens | ||
16. | ALA5191769 | 12g; EML982 | IC50 | = | 4.34 | uM | ALA5138948 | 5.36 | nM | Homo sapiens | ||
17. | ALA5191769 | 12g; EML982 | IC50 | = | 0.778 | uM | ALA5138947 | 6.11 | nM | Homo sapiens | ||
18. | ALA5191769 | 12g; EML982 | IC50 | = | 0.008 | uM | ALA5138946 | 8.08 | nM | Homo sapiens | ||
19. | ALA5191769 | 12g; EML982 | IC50 | = | 13.3 | uM | ALA5138945 | 4.88 | nM | Homo sapiens | ||
20. | ALA5191769 | 12g; EML982 | IC50 | = | 1.8 | uM | ALA5138944 | 5.75 | nM | Homo sapiens |