| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5192384 | 17 | F | = | 16 | % | ALA5160538 | % | ||||
| 2. | ALA5192384 | 17 | F | = | 27 | % | ALA5160537 | % | ||||
| 3. | ALA5192384 | 17 | F | = | 50 | % | ALA5160536 | % | ||||
| 4. | ALA5192384 | 17 | F | = | 62 | % | ALA5160535 | % | ||||
| 5. | ALA5192384 | 17 | t1/2 | = | 43 | hr | ALA5160534 | hr | ||||
| 6. | ALA5192384 | 17 | t1/2 | = | 7.4 | hr | ALA5160533 | hr | ||||
| 7. | ALA5192384 | 17 | CL | = | 1 | ml/min.kg | ALA5160532 | mL.min-1.kg-1 | ||||
| 8. | ALA5192384 | 17 | CL | = | 10.6 | ml/min.kg | ALA5160531 | mL.min-1.kg-1 | ||||
| 9. | ALA5192384 | 17 | IC50 | = | 8.3 | uM | ALA5160530 | 5.08 | nM | |||
| 10. | ALA5192384 | 17 | IC50 | = | 40 | uM | ALA5160529 | 4.40 | nM | |||
| 11. | ALA5192384 | 17 | IC50 | = | 12 | uM | ALA5160528 | 4.92 | nM | |||
| 12. | ALA5192384 | 17 | Activity | 0 | ALA5160527 | Dde | Mus musculus | |||||
| 13. | ALA5192384 | 17 | Activity | 0 | ALA5160526 | Dde | Mus musculus | |||||
| 14. | ALA5192384 | 17 | t1/2 | = | 153 | min | ALA5160525 | hr | Homo sapiens | |||
| 15. | ALA5192384 | 17 | K | = | 4.54 | 10^-3/s | ALA5160524 | 10^-3/s | Homo sapiens | |||
| 16. | ALA5192384 | 17 | Ki | = | 0.11 | nM | ALA5160523 | 9.96 | nM | Homo sapiens | ||
| 17. | ALA5192384 | 17 | IC50 | = | 8643 | nM | ALA5160521 | 5.06 | nM | Homo sapiens | ||
| 18. | ALA5192384 | 17 | CL free | = | 12 | ml/min.kg | ALA5160517 | mL.min-1.kg-1 | ||||
| 19. | ALA5192384 | 17 | CL free | = | 11 | ml/min.kg | ALA5160516 | mL.min-1.kg-1 | ||||
| 20. | ALA5192384 | 17 | solubility | = | 123 | uM | ALA5160515 | nM |
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