| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5192803 | 9c | IC50 | > | 5 | uM | ALA5156610 | nM | Homo sapiens | |||
| 2. | ALA5192803 | 9c | IC50 | = | 0.36 | uM | ALA5156609 | 6.44 | nM | Homo sapiens | ||
| 3. | ALA5192803 | 9c | Drug recovery | = | 95.8 | % | ALA5156608 | % | ||||
| 4. | ALA5192803 | 9c | Drug recovery | = | 106.9 | % | ALA5156607 | % | ||||
| 5. | ALA5192803 | 9c | Ratio | = | 14.17 | ALA5156606 | ||||||
| 6. | ALA5192803 | 9c | Papp | = | 2.89 | 10^-6 cm/s | ALA5156605 | 10^-6 cm/s | ||||
| 7. | ALA5192803 | 9c | Papp | = | 0.2 | 10^-6 cm/s | ALA5156604 | 10^-6 cm/s | ||||
| 8. | ALA5192803 | 9c | ERH | = | 75.35 | % | ALA5156603 | % | ||||
| 9. | ALA5192803 | 9c | ERH | = | 64.03 | % | ALA5156602 | % | ||||
| 10. | ALA5192803 | 9c | CLH | = | 15.6 | ml/min.kg | ALA5156601 | mL.min-1.kg-1 | ||||
| 11. | ALA5192803 | 9c | CLH | = | 35.34 | ml/min.kg | ALA5156600 | mL.min-1.kg-1 | ||||
| 12. | ALA5192803 | 9c | CLH | = | 98.24 | ml/min.kg | ALA5156599 | mL.min-1.kg-1 | ||||
| 13. | ALA5192803 | 9c | CLH | = | 63.27 | ml/min.kg | ALA5156598 | mL.min-1.kg-1 | ||||
| 14. | ALA5192803 | 9c | t1/2 | = | 17.69 | min | ALA5156597 | hr | ||||
| 15. | ALA5192803 | 9c | t1/2 | = | 39.26 | min | ALA5156596 | hr | ||||
| 16. | ALA5192803 | 9c | Stability | = | 16.9 | % | ALA5156595 | % | ||||
| 17. | ALA5192803 | 9c | deltaTm | = | 1.5 | degrees C | ALA5156585 | degrees C | Homo sapiens | |||
| 18. | ALA5192803 | 9c | deltaTm | = | -0.3 | degrees C | ALA5156584 | degrees C | Homo sapiens | |||
| 19. | ALA5192803 | 9c | deltaTm | = | -3 | degrees C | ALA5156583 | degrees C | Homo sapiens | |||
| 20. | ALA5192803 | 9c | deltaTm | = | -0.5 | degrees C | ALA5156582 | degrees C | Homo sapiens |
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