| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5193821 | 29 | Activity | 0 | ALA5142048 | Non-Toxic | ||||||
| 2. | ALA5193821 | 29 | TGI | = | 79 | % | ALA5142046 | % | Homo sapiens | |||
| 3. | ALA5193821 | 29 | TGI | = | 76 | % | ALA5142045 | % | Homo sapiens | |||
| 4. | ALA5193821 | 29 | TGI | = | 71 | % | ALA5142044 | % | Homo sapiens | |||
| 5. | ALA5193821 | 29 | F | = | 110 | % | ALA5142041 | % | ||||
| 6. | ALA5193821 | 29 | F | = | 106 | % | ALA5142040 | % | ||||
| 7. | ALA5193821 | 29 | AUC | = | 25046 | hr.ng/ml | ALA5142039 | ng.hr.mL-1 | ||||
| 8. | ALA5193821 | 29 | AUC | = | 23807 | hr.ng/ml | ALA5142038 | ng.hr.mL-1 | ||||
| 9. | ALA5193821 | 29 | Tmax | = | 1 | hr | ALA5142037 | hr | ||||
| 10. | ALA5193821 | 29 | Tmax | = | 4 | hr | ALA5142036 | hr | ||||
| 11. | ALA5193821 | 29 | Cmax | = | 3810 | ng/ml | ALA5142035 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 12. | ALA5193821 | 29 | Cmax | = | 2193 | ng/ml | ALA5142034 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 13. | ALA5193821 | 29 | t1/2 | = | 5 | hr | ALA5142033 | hr | ||||
| 14. | ALA5193821 | 29 | t1/2 | = | 4 | hr | ALA5142032 | hr | ||||
| 15. | ALA5193821 | 29 | Vdss | = | 2.4 | L/Kg | ALA5142031 | L.kg-1 | ||||
| 16. | ALA5193821 | 29 | Vdss | = | 2.2 | L/Kg | ALA5142030 | L.kg-1 | ||||
| 17. | ALA5193821 | 29 | CL | = | 7.3 | ml/min.kg | ALA5142029 | mL.min-1.kg-1 | ||||
| 18. | ALA5193821 | 29 | CL | = | 7.6 | ml/min.kg | ALA5142028 | mL.min-1.kg-1 | ||||
| 19. | ALA5193821 | 29 | IC50 | > | 10 | uM | ALA5142027 | nM | Homo sapiens | |||
| 20. | ALA5193821 | 29 | IC50 | > | 10 | uM | ALA5142026 | nM | Homo sapiens |
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