| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5194984 | 1 | Vdss | = | 1.31 | L/Kg | ALA5159679 | L.kg-1 | ||||
| 2. | ALA5194984 | 1 | F | = | 15.7 | % | ALA5159678 | % | ||||
| 3. | ALA5194984 | 1 | MRT | = | 4.05 | hr | ALA5159677 | hr | ||||
| 4. | ALA5194984 | 1 | CL | = | 1.42 | L/hr/kg | ALA5159676 | mL.min-1.kg-1 | ||||
| 5. | ALA5194984 | 1 | t1/2 | = | 1.14 | hr | ALA5159675 | hr | ||||
| 6. | ALA5194984 | 1 | t1/2 | = | 1.62 | hr | ALA5159674 | hr | ||||
| 7. | ALA5194984 | 1 | AUC | = | 1422 | ng.hr/ml | ALA5159673 | ng.hr.mL-1 | ||||
| 8. | ALA5194984 | 1 | AUC | = | 562 | ng.hr/ml | ALA5159672 | ng.hr.mL-1 | ||||
| 9. | ALA5194984 | 1 | MRT | = | 0.932 | hr | ALA5159671 | hr | ||||
| 10. | ALA5194984 | 1 | Cmax | = | 192 | ng/ml | ALA5159670 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 11. | ALA5194984 | 1 | Tmax | = | 1.67 | hr | ALA5159669 | hr | ||||
| 12. | ALA5194984 | 1 | IC50 | = | 454 | nM | ALA5159665 | 6.34 | nM | Mus musculus | ||
| 13. | ALA5194984 | 1 | IC50 | = | 413 | nM | ALA5159664 | 6.38 | nM | Homo sapiens | ||
| 14. | ALA5194984 | 1 | IC50 | = | 118 | nM | ALA5159663 | 6.93 | nM | Homo sapiens | ||
| 15. | ALA5194984 | 1 | IC50 | = | 0.075 | uM | ALA5159662 | 7.13 | nM | Homo sapiens |
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