| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5195440 | 7 | F | = | 60 | % | ALA5125593 | % | ||||
| 2. | ALA5195440 | 7 | t1/2 | = | 2.7 | hr | ALA5125592 | hr | ||||
| 3. | ALA5195440 | 7 | AUC | = | 7.7 | ug.hr/ml | ALA5125591 | ng.hr.mL-1 | ||||
| 4. | ALA5195440 | 7 | Cmax | = | 1.6 | ug ml-1 | ALA5125590 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 5. | ALA5195440 | 7 | t1/2 | = | 4.1 | hr | ALA5125589 | hr | ||||
| 6. | ALA5195440 | 7 | AUC | = | 1.3 | ug.hr/ml | ALA5125588 | ng.hr.mL-1 | ||||
| 7. | ALA5195440 | 7 | Vdss | = | 2.7 | L/Kg | ALA5125587 | L.kg-1 | ||||
| 8. | ALA5195440 | 7 | CL | = | 14 | ml/min.kg | ALA5125586 | mL.min-1.kg-1 | ||||
| 9. | ALA5195440 | 7 | F | = | 55 | % | ALA5125581 | % | ||||
| 10. | ALA5195440 | 7 | t1/2 | = | 0.8 | hr | ALA5125580 | hr | ||||
| 11. | ALA5195440 | 7 | AUC | = | 14 | ug.hr/ml | ALA5125579 | ng.hr.mL-1 | ||||
| 12. | ALA5195440 | 7 | Cmax | = | 7.6 | ug ml-1 | ALA5125578 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM | |||
| 13. | ALA5195440 | 7 | t1/2 | = | 1.6 | hr | ALA5125577 | hr | ||||
| 14. | ALA5195440 | 7 | AUC | = | 0.5 | ug.hr/ml | ALA5125576 | ng.hr.mL-1 | ||||
| 15. | ALA5195440 | 7 | Vdss | = | 2.9 | L/Kg | ALA5125575 | L.kg-1 | ||||
| 16. | ALA5195440 | 7 | CL | = | 35 | ml/min.kg | ALA5125574 | mL.min-1.kg-1 | ||||
| 17. | ALA5195440 | 7 | IC50 | > | 25 | uM | ALA5125559 | nM | Homo sapiens | |||
| 18. | ALA5195440 | 7 | IC50 | = | 10.8 | uM | ALA5125558 | 4.97 | nM | Homo sapiens | ||
| 19. | ALA5195440 | 7 | IC50 | > | 25 | uM | ALA5125557 | nM | Homo sapiens | |||
| 20. | ALA5195440 | 7 | IC50 | > | 25 | uM | ALA5125556 | nM | Homo sapiens |
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