| # | Name | Compound Key | Action Type | Relation | Activity Value | Units | Assay ID | Assay Description | Comment | Assay | Assay Organism | |
|---|---|---|---|---|---|---|---|---|---|---|---|---|
| 1. |  ALA5196874 | (-)-53; MU1656 | Stability | = | 41 | % | ALA5162127 | % | ||||
| 2. | ALA5196874 | (-)-53; MU1656 | CLH | = | 56 | microL/min/mg | ALA5162126 | mL.min-1.g-1 | ||||
| 3. | ALA5196874 | (-)-53; MU1656 | Activity | 0 | ALA5162125 | Non-Toxic | ||||||
| 4. | ALA5196874 | (-)-53; MU1656 | F | 0 | ALA5162120 | ND | % | |||||
| 5. | ALA5196874 | (-)-53; MU1656 | CL | = | 14.2 | ml/min.kg | ALA5162118 | mL.min-1.kg-1 | ||||
| 6. | ALA5196874 | (-)-53; MU1656 | CL | = | 9.54 | ml/min.kg | ALA5162117 | mL.min-1.kg-1 | ||||
| 7. | ALA5196874 | (-)-53; MU1656 | Vd | = | 1180 | ml/kg | ALA5162116 | L.kg-1 | ||||
| 8. | ALA5196874 | (-)-53; MU1656 | Vd | 0 | ALA5162115 | ND | ||||||
| 9. | ALA5196874 | (-)-53; MU1656 | Vd | = | 1290 | ml/kg | ALA5162114 | L.kg-1 | ||||
| 10. | ALA5196874 | (-)-53; MU1656 | Kel | = | 0.012 | /min | ALA5162113 | /min | ||||
| 11. | ALA5196874 | (-)-53; MU1656 | Kel | 0 | ALA5162112 | ND | ||||||
| 12. | ALA5196874 | (-)-53; MU1656 | Kel | = | 0.007 | /min | ALA5162111 | /min | ||||
| 13. | ALA5196874 | (-)-53; MU1656 | t1/2 | = | 57.2 | min | ALA5162110 | hr | ||||
| 14. | ALA5196874 | (-)-53; MU1656 | t1/2 | 0 | ALA5162109 | ND | ||||||
| 15. | ALA5196874 | (-)-53; MU1656 | t1/2 | = | 93.6 | min | ALA5162108 | hr | ||||
| 16. | ALA5196874 | (-)-53; MU1656 | AUC | = | 351000 | ng.min/ml | ALA5162107 | ng.hr.mL-1 | ||||
| 17. | ALA5196874 | (-)-53; MU1656 | AUC | = | 2100000 | ng.min/ml | ALA5162105 | ng.hr.mL-1 | ||||
| 18. | ALA5196874 | (-)-53; MU1656 | AUCt | = | 348000 | ng.min/ml | ALA5162104 | ng.hr.mL-1 | ||||
| 19. | ALA5196874 | (-)-53; MU1656 | AUCt | = | 2080000 | ng.min/ml | ALA5162102 | ng.hr.mL-1 | ||||
| 20. | ALA5196874 | (-)-53; MU1656 | Cmax | = | 20600 | ng/ml | ALA5162101 | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | standard_value was converted from ug.mL-1 to nM using the parent compound MW | nM |
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